SCHEMBL26019477

SCHEMBL26019477

O=C(ON1C[C@H]2C[C@H](O)C[C@H]2C1)c1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
F2 P00734 1/20 0.41
LMNA P02545 1/20 0.41
CHRNA7 P36544 5/20 0.40
HTR3E A5X5Y0 1/20 0.40
HTR3B O95264 1/20 0.40
HTR3A P46098 1/20 0.40
HTR3D Q70Z44 1/20 0.40
HTR3C Q8WXA8 1/20 0.40
TSHR P16473 2/20 0.40
KMT2A Q03164 2/20 0.40
PIK3CD O00329 1/20 0.39
MEN1 O00255 1/20 0.38
GRIN2B Q13224 1/20 0.38
CHRNB2 P17787 2/20 0.38
CHRNA4 P43681 2/20 0.38
CHRNA5 P30532 1/20 0.38
NPC1 O15118 1/20 0.37
CHRNB4 P30926 1/20 0.37
CHRNA3 P32297 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26018931 1.00 F2 (0.41) F2LMNACHRNA7HTR3EHTR3B
SCHEMBL25796422 0.86 F2 (0.47) F2LMNACHRNA7HTR3EHTR3B
SCHEMBL26497408 0.82 HTR3E (0.43) F2LMNACHRNA7HTR3EHTR3B
SCHEMBL26019479 0.82 CHRNA7 (0.40) CHRNA7HTR3EHTR3BHTR3AHTR3D
SCHEMBL26019255 0.82 CHRNA7 (0.40) CHRNA7HTR3EHTR3BHTR3AHTR3D
SCHEMBL29346476 0.82 CHRNA7 (0.40) CHRNA7HTR3EHTR3BHTR3AHTR3D
SCHEMBL11061761 0.78 TSHR (0.47) F2LMNACHRNA7HTR3EHTR3B
SCHEMBL26545466 0.78 F2 (0.45) F2LMNACHRNA7HTR3EHTR3B
SCHEMBL25845894 0.78 F2 (0.45) F2LMNACHRNA7HTR3EHTR3B
SCHEMBL28781857 0.77 KMT2A (0.44) F2LMNACHRNA7HTR3EHTR3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3974420-B1 N-ALKYLARYL-5-OXYHETEROARYL-OCTAHYDRO-CYCLOPENTA[C]PYRROLE NEGATIVE ALLOSTERIC MODULATORS OF NR2B NOVARTIS AG (CH) 2023-08-16 EP disclosed