SCHEMBL26041260

SCHEMBL26041260

CCCCCC(=O)N(C)Cc1cc(-c2ncco2)ccc1-c1ccccc1S(=O)(=O)Nc1noc(C)c1C

nearest known ligand 0.80

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
EDNRA P25101 16/20 0.80
EDNRB P24530 19/20 0.67

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6641356 0.91 EDNRA (0.86) EDNRAEDNRB
Edonentan SCHEMBL29742313 0.89 EDNRA (1.00) EDNRAEDNRB
Edonentan SCHEMBL1651069 0.89 EDNRA (1.00) EDNRAEDNRB
SCHEMBL6638555 0.82 EDNRB (0.92) EDNRAEDNRB
SCHEMBL6703895 0.82 EDNRA (0.71) EDNRAEDNRB
SCHEMBL26552022 0.81 EDNRA (0.76) EDNRAEDNRB
SCHEMBL6642915 0.80 EDNRB (0.79) EDNRAEDNRB
SCHEMBL6642249 0.80 EDNRB (1.00) EDNRAEDNRB
SCHEMBL6963011 0.79 EDNRA (0.68) EDNRAEDNRB
SCHEMBL6641551 0.79 EDNRB (0.83) EDNRAEDNRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11738007-B2 Treatment of glaucoma using endothelin receptor antagonists PERFUSE THERAPEUTICS, INC. (US) 2023-08-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11738007-B2 Treatment of glaucoma using endothelin receptor antagonists EDNRA, EDNRB, FLT1 EDNRA 1/4885EDNRB 2/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.