SCHEMBL260523

SCHEMBL260523

Cc1ccc(-c2ccc(CN=C=O)cc2)cc1

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.38
C3AR1 Q16581 1/20 0.38
HRH3 Q9Y5N1 2/20 0.37
FFAR1 O14842 1/20 0.37
S1PR1 P21453 1/20 0.37
S1PR5 Q9H228 1/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
NAAA Q02083 2/20 0.36
MIF P14174 2/20 0.36
PYCR1 P32322 1/20 0.36
CYP1A2 P05177 1/20 0.35
CYP2A6 P11509 1/20 0.35
TAAR1 Q96RJ0 1/20 0.35
TRPA1 O75762 1/20 0.35
CTBP2 P56545 1/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL436823 0.94 IDO1 (0.42) IDO1C3AR1FFAR1MIFPYCR1
SCHEMBL21089 0.84 MIF (0.44) MIFCYP1A2TRPA1
SCHEMBL4600494 0.83 ALDH1A1 (0.47) IDO1FFAR1MEN1KMT2ANAAA
Toluene SCHEMBL28728282 0.83 MIF (0.47) C3AR1MEN1KMT2AMIFTRPA1
Water SCHEMBL14972874 0.82 MIF (0.43) MIFTRPA1
SCHEMBL22471901 0.82 MIF (0.43) MIFTRPA1
Water SCHEMBL29040332 0.82 MIF (0.43) MIFTRPA1
SCHEMBL12885577 0.82 C3AR1 (0.37) IDO1C3AR1S1PR1S1PR5MEN1
Water SCHEMBL27998963 0.82 ALDH1A1 (0.45) IDO1FFAR1MEN1KMT2ANAAA
SCHEMBL9716383 0.80 CYP3A4 (0.59) HRH3MIFCYP1A2TRPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8067440-B2 Phosphonium salts derivatives and uses thereof VALORISATION-RECHERCHE, LIMITED PARTNERSHIP (CA) 2011-11-29 US disclosed
US-20110092683-A1 PHOSPHONIUM SALTS DERIVATIVES AND USES THEREOF VALORISATION-RECHERCHE, LIMITED PARTNERSHIP (CA) 2011-04-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110092683-A1 PHOSPHONIUM SALTS DERIVATIVES AND USES THEREOF PI4K2A, PIP4K2A, PI4K2B IDO1 3934/4885C3AR1 1632/4885HRH3 3748/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.