SCHEMBL26062928

SCHEMBL26062928

COc1ccc(C2CCCCC2)c2ncc(C)nc12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.40
NPC1 O15118 1/20 0.40
ALDH1A1 P00352 1/20 0.40
HPGD P15428 1/20 0.40
RAB9A P51151 1/20 0.40
HSD17B10 Q99714 1/20 0.40
CDK4 P11802 3/20 0.40
CCND1 P24385 3/20 0.40
CDK1 P06493 1/20 0.40
CCNB1 P14635 1/20 0.40
CCNE1 P24864 1/20 0.40
CDK2 P24941 1/20 0.40
PDGFRB P09619 5/20 0.40
PDGFRA P16234 5/20 0.40
PDK2 Q15119 1/20 0.39
PDK4 Q16654 1/20 0.39
MAPT P10636 1/20 0.39
PTGDR2 Q9Y5Y4 2/20 0.38
NQO2 P16083 1/20 0.37
PDE10A Q9Y233 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26063528 0.87 ADORA2A (0.41) CDK4CCND1CDK1CCNB1CCNE1
SCHEMBL13313319 0.79 MAPT (0.52) KDM4ENPC1ALDH1A1HPGDRAB9A
SCHEMBL26063053 0.78 MAPT (0.51) ALDH1A1HSD17B10PDGFRBPDGFRAMAPT
SCHEMBL20867659 0.75 KDM4E (0.45) KDM4ENPC1ALDH1A1HPGDHSD17B10
SCHEMBL20765414 0.75 ADORA2A (0.40) ALDH1A1CDK4CCND1CDK1CCNB1
SCHEMBL20764935 0.74 ADORA2A (0.39) CDK4CCND1CDK1CCNB1CCNE1
SCHEMBL30439753 0.74 ADORA2A (0.39) CDK4CCND1CDK1CCNB1CCNE1
SCHEMBL5581664 0.72 CDK4 (0.46) KDM4ENPC1ALDH1A1HPGDRAB9A
SCHEMBL26045395 0.72 ALDH1A1 (0.49) KDM4ENPC1ALDH1A1HPGDRAB9A
SCHEMBL20764934 0.70 ADORA2A (0.42) PDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3672951-B1 QUINOXALINE DERIVATIVES AS ADENOSINE RECEPTOR ANTAGONISTS MERCK PATENT GMBH (DE) 2023-08-30 EP disclosed