SCHEMBL26063993

SCHEMBL26063993

CS(=O)(=O)CCn1cc(CN)nn1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CA12 O43570 2/20 0.41
CA1 P00915 2/20 0.41
CA2 P00918 2/20 0.41
CA9 Q16790 2/20 0.41
NOTUM Q6P988 3/20 0.38
MAOA P21397 4/20 0.37
MAOB P27338 2/20 0.35
LOXL2 Q9Y4K0 4/20 0.34
GGPS1 O95749 2/20 0.33
HSP90AB1 P08238 1/20 0.32
KDM1A O60341 1/20 0.32
PTGS2 P35354 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25356726 0.83 NOTUM (0.34) NOTUMHSP90AB1KDM1APTGS2
SCHEMBL25357577 0.83 NOTUM (0.44) CA12CA1CA2CA9NOTUM
SCHEMBL26036597 0.83 HSP90AB1 (0.35) NOTUMHSP90AB1
Hydrochloric Acid SCHEMBL25355887 0.82 NOTUM (0.33) NOTUMLOXL2HSP90AB1KDM1APTGS2
SCHEMBL25416332 0.76 CA12 (0.41) CA12CA1CA2CA9NOTUM
SCHEMBL26066624 0.76 CA12 (0.39) CA12CA1CA2CA9NOTUM
SCHEMBL28174204 0.74 NOTUM (0.43) CA12CA1CA2CA9NOTUM
SCHEMBL12825274 0.74 GBA1 (0.48)
SCHEMBL24345690 0.73 P2RX7 (0.38)
SCHEMBL26066626 0.73 HRH4 (0.38) CA12CA1CA2CA9NOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023154344-A1 2-METHYL-4',5'-DIHYDROSPIRO[PIPERIDINE-4,7'-THIENO[2,3-C]PYRAN] DERIVATIVES AS INHIBITORS OF APOL1 AND METHODS OF USING SAME VERTEX PHARMACEUTICALS INCORPORATED (US) 2023-08-17 WO disclosed