SCHEMBL2609237

SCHEMBL2609237

Cc1cc(N2C[C@H](Cc3ccc(OCC(F)(F)F)cc3Cl)C[C@H]2C(=O)NC2(C#N)CC2)n(C2CCC2)n1

nearest known ligand 0.47

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CTSS P25774 20/20 0.47
CTSL P07711 16/20 0.47
CTSK P43235 3/20 0.39
CTSB P07858 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL701451 0.88 CTSS (0.61) CTSSCTSLCTSKCTSB
SCHEMBL696153 0.84 CTSS (0.54) CTSSCTSLCTSKCTSB
SCHEMBL696411 0.84 CTSS (0.54) CTSSCTSLCTSKCTSB
SCHEMBL696432 0.83 CTSS (0.60) CTSSCTSLCTSK
SCHEMBL695203 0.83 CTSS (0.60) CTSSCTSLCTSK
SCHEMBL15338583 0.81 CTSS (0.39) CTSSCTSLCTSKCTSB
SCHEMBL15327207 0.80 CTSS (0.53) CTSSCTSLCTSKCTSB
SCHEMBL2106860 0.78 CTSS (0.51) CTSSCTSLCTSKCTSB
SCHEMBL694369 0.78 CTSS (0.58) CTSSCTSLCTSKCTSB
SCHEMBL2609235 0.77 CTSS (0.42) CTSSCTSLCTSKCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8163793-B2 Proline derivatives HOFFMAN-LA ROCHE INC. (US) 2012-04-24 US disclosed