SCHEMBL26148387

SCHEMBL26148387

O=C(Cc1ccccc1)NCc1ccc2c(c1)CN(C1CCC(=O)NC1=O)C2=O

nearest known ligand 0.63

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CRBN Q96SW2 12/20 0.63
DDB1 Q16531 4/20 0.63
GSPT1 P15170 2/20 0.63
CYP2C19 P33261 1/20 0.63
KCNH2 Q12809 1/20 0.63
IKZF3 Q9UKT9 2/20 0.62
CSNK1A1 P48729 2/20 0.60
IKZF2 Q9UKS7 6/20 0.59
IKZF1 Q13422 1/20 0.54
MAP1LC3B Q9GZQ8 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1403628 0.92 CRBN (0.66) CRBNDDB1GSPT1CYP2C19KCNH2
SCHEMBL26148525 0.92 CRBN (0.64) CRBNDDB1GSPT1CYP2C19KCNH2
SCHEMBL1413563 0.92 CRBN (0.74) CRBNDDB1GSPT1CYP2C19KCNH2
SCHEMBL13578966 0.92 CRBN (0.62) CRBNDDB1GSPT1CYP2C19KCNH2
SCHEMBL1403675 0.92 CRBN (0.62) CRBNDDB1GSPT1CYP2C19KCNH2
SCHEMBL26148713 0.91 CRBN (0.61) CRBNDDB1GSPT1CYP2C19KCNH2
SCHEMBL1403669 0.90 CRBN (0.65) CRBNDDB1GSPT1CYP2C19KCNH2
SCHEMBL1403618 0.90 CRBN (0.62) CRBNDDB1GSPT1CYP2C19KCNH2
SCHEMBL16381535 0.90 CRBN (0.62) CRBNDDB1GSPT1CYP2C19KCNH2
SCHEMBL15841617 0.90 CRBN (0.62) CRBNDDB1GSPT1CYP2C19KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118201917-A Compound with degradation GSPT1 activity and application thereof 上海美志医药科技有限公司 2024-06-14 CN disclosed
WO-2023078410-A1 COMPOUND HAVING ACTIVITY OF DEGRADING GSPT1 AND APPLICATION THEREOF 上海美志医药科技有限公司 2023-05-11 WO disclosed
WO-2023078410-A1 COMPOUND HAVING ACTIVITY OF DEGRADING GSPT1 AND APPLICATION THEREOF 上海美志医药科技有限公司 2023-05-11 WO disclosed
CN-116082301-A Compound with GSPT1 degradation activity and application thereof 上海美志医药科技有限公司 2023-05-09 CN disclosed