SCHEMBL26176201

SCHEMBL26176201

CN1CCN(c2cccc(Nc3ccc4c(-c5ccc6nccn6n5)c[nH]c4n3)c2)CC1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 7/20 0.56
FLT3 P36888 5/20 0.56
CCNE1 P24864 3/20 0.56
CDK1 P06493 2/20 0.56
CCNB1 P14635 2/20 0.56
CDK7 P50613 2/20 0.56
CCNH P51946 2/20 0.56
MNAT1 P51948 2/20 0.56
DYRK1B Q9Y463 2/20 0.41
IGF1R P08069 1/20 0.41
JAK2 O60674 10/20 0.40
JAK3 P52333 10/20 0.40
PTK2 Q05397 9/20 0.40
CCNT1 O60563 1/20 0.40
CCNA2 P20248 1/20 0.40
CDK9 P50750 1/20 0.40
EGFR P00533 1/20 0.40
PRKCI P41743 1/20 0.39
WEE1 P30291 1/20 0.38
ABCB1 P08183 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30399350 1.00 CDK2 (0.56) CDK2FLT3CCNE1CDK1CCNB1
SCHEMBL25157783 0.88 CDK2 (0.59) CDK2FLT3CCNE1CDK1CCNB1
SCHEMBL30346738 0.88 CDK2 (0.59) CDK2FLT3CCNE1CDK1CCNB1
SCHEMBL30399447 0.83 FLT3 (0.51) CDK2FLT3CCNE1CDK1CCNB1
SCHEMBL26176191 0.83 FLT3 (0.51) CDK2FLT3CCNE1CDK1CCNB1
SCHEMBL30399648 0.80 FLT3 (0.49) CDK2FLT3CCNE1CDK1CCNB1
SCHEMBL26176198 0.80 FLT3 (0.49) CDK2FLT3CCNE1CDK1CCNB1
SCHEMBL30400250 0.78 CDK2 (0.57) CDK2FLT3CCNE1CDK1CCNB1
SCHEMBL26176213 0.78 CDK2 (0.57) CDK2FLT3CCNE1CDK1CCNB1
SCHEMBL30399562 0.78 CDK2 (0.49) CDK2FLT3CCNE1CDK1CCNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230192686-A1 1H-PYRROLO[2,3-B]PYRIDINES AND PREPARATION AND USES THEREOF TENARX, INC. 2023-06-22 US disclosed
US-20230192686-A1 1H-PYRROLO[2,3-B]PYRIDINES AND PREPARATION AND USES THEREOF TENARX, INC. 2023-06-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230192686-A1 1H-PYRROLO[2,3-B]PYRIDINES AND PREPARATION AND USES THEREOF DYRK1A, DYRK1B, DYRK2 CDK2 212/4885FLT3 1398/4885CCNE1 1178/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.