SCHEMBL2623243

SCHEMBL2623243

[3H]c1cccc(-c2ccc(N(c3ccccc3)c3ccc(OCCCCCCCOc4ccc(N(c5ccccc5)c5ccc(-c6cccc([3H])c6)cc5)cc4)cc3)cc2)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LSS P48449 1/20 0.49
HDAC3 O15379 9/20 0.48
HDAC4 P56524 9/20 0.48
HDAC1 Q13547 9/20 0.48
HDAC7 Q8WUI4 9/20 0.48
HDAC2 Q92769 9/20 0.48
HDAC10 Q969S8 9/20 0.48
HDAC11 Q96DB2 9/20 0.48
HDAC8 Q9BY41 9/20 0.48
HDAC6 Q9UBN7 9/20 0.48
HDAC9 Q9UKV0 9/20 0.48
HDAC5 Q9UQL6 9/20 0.48
HRH3 Q9Y5N1 5/20 0.46
KCNH2 Q12809 1/20 0.46
HRH4 Q9H3N8 1/20 0.46
CHRNB2 P17787 1/20 0.43
CHRNB4 P30926 1/20 0.43
CHRNA3 P32297 1/20 0.43
CHRNA7 P36544 1/20 0.43
CHRNA4 P43681 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2623368 0.86 LSS (0.49) LSSHDAC3HDAC4HDAC1HDAC7
SCHEMBL2623380 0.85 RARB (0.43) LSSHDAC3HDAC4HDAC1HDAC7
SCHEMBL2623299 0.85 HRH3 (0.46) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL2623356 0.84 KCNA3 (0.42) LSSHRH3CHRNB2CHRNB4CHRNA3
SCHEMBL8943680 0.84 KCNA3 (0.60) LSSHDAC3HDAC4HDAC1HDAC7
SCHEMBL8943908 0.84 KCNA3 (0.60) LSSHDAC3HDAC4HDAC1HDAC7
SCHEMBL8944087 0.84 KCNA3 (0.60) LSSHDAC3HDAC4HDAC1HDAC7
SCHEMBL8944286 0.84 KCNA3 (0.60) LSSHDAC3HDAC4HDAC1HDAC7
SCHEMBL12972985 0.83 LTA4H (0.60) LSSHRH3KCNH2
SCHEMBL22770745 0.83 LTA4H (0.60) LSSHRH3KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120091443-A1 COMPOSITION FOR USE IN ORGANIC DEVICE, POLYMER FILM, AND ORGANIC ELECTROLUMINESCENT ELEMENT MITSUBISHI CHEMICAL CORPORATION (JP) 2012-04-19 US disclosed
US-20100045174-A1 COMPOSITION FOR USE IN ORGANIC DEVICE, POLYMER FILM, AND ORGANIC ELECTROLUMINESCENT ELEMENT MITSUBISHI CHEMICAL CORPORATION (JP) 2010-02-25 US disclosed