SCHEMBL26242535

SCHEMBL26242535

Cc1nnc(-c2cccnc2)c(C)c1C

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 12/20 0.53
CYP3A4 P08684 6/20 0.50
ALDH1A1 P00352 2/20 0.50
CYP1A2 P05177 1/20 0.50
KDM4E B2RXH2 1/20 0.48
LMNA P02545 1/20 0.48
TP53 P04637 1/20 0.48
MAPT P10636 1/20 0.48
HPGD P15428 1/20 0.48
ALOX15 P16050 1/20 0.48
HTT P42858 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
HSD17B10 Q99714 1/20 0.48
CYP2C9 P11712 4/20 0.46
CYP2B6 P20813 4/20 0.46
CYP2E1 P05181 3/20 0.46
CYP2C19 P33261 3/20 0.46
CYP2D6 P10635 2/20 0.46
NPY5R Q15761 1/20 0.45
MAP2K4 P45985 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26242505 0.78 MAOB (0.44) ALDH1A1KDM4EMAPTHPGDSMN1; SMN2
SCHEMBL26242537 0.78 MAPT (0.43) ALDH1A1CYP1A2KDM4ELMNATP53
SCHEMBL30385344 0.74 CYP2A6 (0.49) CYP2A6CYP3A4ALDH1A1CYP1A2KDM4E
SCHEMBL18818721 0.73 CYP2A6 (0.67) CYP2A6CYP3A4ALDH1A1CYP1A2KDM4E
SCHEMBL13910994 0.71 CYP2A6 (0.70) CYP2A6CYP3A4ALDH1A1CYP1A2KDM4E
SCHEMBL28058405 0.70 CYP2A6 (0.53) CYP2A6CYP3A4ALDH1A1CYP1A2KDM4E
SCHEMBL5931880 0.70 CYP2A6 (0.53) CYP2A6CYP3A4ALDH1A1CYP1A2KDM4E
SCHEMBL16826037 0.70 CYP2A6 (0.53) CYP2A6CYP3A4ALDH1A1CYP1A2KDM4E
SCHEMBL9807161 0.70 NPSR1 (0.61) CYP2A6CYP3A4ALDH1A1KDM4ELMNA
SCHEMBL26242506 0.70 CNR1 (0.45) ALDH1A1KDM4ELMNAMAPTALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023150201-A2 SODIUM CHANNEL BLOCKING COMPOUNDS, DERIVATIVES THEREOF, AND METHODS OF THEIR USE LATIGO BIOTHERAPEUTICS, INC. (US) 2023-08-10 WO disclosed