SCHEMBL2625575

SCHEMBL2625575

CC(C)Nc1nn(C)c(=O)[nH]1

nearest known ligand 0.37

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
KAT2B Q92831 1/20 0.35
ATM Q13315 1/20 0.34
CSNK2A2 P19784 1/20 0.33
CSNK2B P67870 1/20 0.33
CSNK2A1 P68400 1/20 0.33
HTT P42858 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8368738 0.77
SCHEMBL20848461 0.64 TSHR (0.42) KDM4EALDH1A1CSNK2A2CSNK2BCSNK2A1
SCHEMBL9980116 0.63 ATM (0.33) ATM
SCHEMBL6767648 0.63 ATM (0.36) ATM
SCHEMBL10105029 0.61 GRIA1 (0.42) KDM4EALDH1A1ATM
SCHEMBL22743552 0.60 DAO (0.34) ATM
SCHEMBL16131591 0.60 GRIA1 (0.41) ATM
SCHEMBL7762067 0.60 ATM (0.37) ATM
SCHEMBL15563493 0.60 DAO (0.38) ATM
SCHEMBL12702610 0.60 DAO (0.38) ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8163763-B2 Pyrimidine compounds, compositions and methods of use GENENTECH, INC. (US) 2012-04-24 US disclosed
US-8163763-B2 Pyrimidine compounds, compositions and methods of use GENENTECH, INC. (US) 2012-04-24 US disclosed