Taribavirin

Taribavirin

SCHEMBL2631656

N=C(N)c1ncn([C@@H]2O[C@H](CO)C(O)C2O)n1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PNP P00491 4/20 1.00
LMNA P02545 4/20 0.76
SMN1; SMN2 Q16637 4/20 0.76
ALDH1A1 P00352 3/20 0.76
TSHR P16473 2/20 0.76
THPO P40225 2/20 0.76
PMP22 Q01453 2/20 0.76
ADORA1 P30542 2/20 0.76
GLA P06280 1/20 0.76
EIF4E P06730 1/20 0.76
CYP3A4 P08684 1/20 0.76
TOP1 P11387 1/20 0.76
KDM4E B2RXH2 2/20 0.47
HTT P42858 2/20 0.47
BLM P54132 2/20 0.47
TP53 P04637 2/20 0.47
MAPT P10636 2/20 0.47
TDP1 Q9NUW8 1/20 0.47
GAA P10253 1/20 0.47
GMNN O75496 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Taribavirin SCHEMBL3868643 1.00 PNP (1.00) PNPLMNASMN1; SMN2ALDH1A1TSHR
Taribavirin SCHEMBL2619250 1.00 PNP (1.00) PNPLMNASMN1; SMN2ALDH1A1TSHR
Taribavirin SCHEMBL12758161 1.00 PNP (1.00) PNPLMNASMN1; SMN2ALDH1A1TSHR
Taribavirin SCHEMBL3307695 1.00 PNP (1.00) PNPLMNASMN1; SMN2ALDH1A1TSHR
Taribavirin SCHEMBL3307685 1.00 PNP (1.00) PNPLMNASMN1; SMN2ALDH1A1TSHR
Taribavirin SCHEMBL4967368 1.00 PNP (1.00) PNPLMNASMN1; SMN2ALDH1A1TSHR
Taribavirin SCHEMBL16330745 1.00 PNP (1.00) PNPLMNASMN1; SMN2ALDH1A1TSHR
Taribavirin SCHEMBL6981526 1.00 PNP (1.00) PNPLMNASMN1; SMN2ALDH1A1TSHR
Taribavirin SCHEMBL18735565 1.00 PNP (1.00) PNPLMNASMN1; SMN2ALDH1A1TSHR
Taribavirin SCHEMBL40670 1.00 PNP (1.00) PNPLMNASMN1; SMN2ALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9828409-B2 Bridged-cyclo-ProTides as prodrugs of therapeutic nucleosides and nucleotides ZHONG MINGHONG (US) 2017-11-28 US disclosed
US-20120101157-A1 4,5-Diamino-3-Halo-2-Hydroxybenzoic Acid Derivatives and Preparations Thereof NATIONAL DEFENSE MEDICAL CENTER (TW) 2012-04-26 US disclosed
WO-2011076923-A9 INHIBITOR FOR INOSINE MONOPHOSPHATE (IMP) DEHYDROGENASE AND/OR VIRAL RNA POLYMERASE FOR TREATMENT OF HEPATITIS E INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (FR) 2011-08-18 WO disclosed
WO-2011076923-A1 INHIBITOR FOR INOSINE MONOPHOSPHATE (IMP) DEHYDROGENASE AND/OR VIRAL RNA POLYMERASE FOR TREATMENT OF HEPATITIS E INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (FR) 2011-06-30 WO disclosed
US-20100298256-A1 ANTIVIRAL COMPOUNDS EPIPHANY BIOSCIENCES, INC. 2010-11-25 US disclosed
US-7816339-B2 Treatments for Flaviviridae virus infection SCHERING CORPORATION (US) 2010-10-19 US disclosed
US-20090209483-A1 TREATMENTS FOR FLAVIVIRIDAE VIRUS INFECTION SCHERING CORPORATION 2009-08-20 US disclosed
WO-2009085267-A1 ANTIVIRAL COMPOUNDS EPIPHANY BIOSCIENCES (US) 2009-07-09 WO disclosed
WO-2008082601-A2 COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS FOR THE TREATMENT OF VIRAL INFECTIONS IDENIX PHARMACEUTICALS, INC. (US) 2008-07-10 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090209483-A1 TREATMENTS FOR FLAVIVIRIDAE VIRUS INFECTION HAVCR2, EIF2AK2, HNRNPC PNP 131/4885LMNA 2114/4885SMN1; SMN2 3971/4885
US-20120101157-A1 4,5-Diamino-3-Halo-2-Hydroxybenzoic Acid Derivatives and Preparations Thereof H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16, HRH3, HRH2 PNP 1819/4885LMNA 3184/4885SMN1; SMN2 4664/4885
US-20100298256-A1 ANTIVIRAL COMPOUNDS MTAP, PNP, TYMP PNP 2/4885LMNA 2760/4885SMN1; SMN2 2573/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.