Taribavirin

Taribavirin

SCHEMBL4967368

N=C(N)c1ncn(C2O[C@H](CO)[C@@H](O)[C@H]2O)n1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PNP P00491 4/20 1.00
LMNA P02545 4/20 0.76
SMN1; SMN2 Q16637 4/20 0.76
ALDH1A1 P00352 3/20 0.76
TSHR P16473 2/20 0.76
THPO P40225 2/20 0.76
PMP22 Q01453 2/20 0.76
ADORA1 P30542 2/20 0.76
GLA P06280 1/20 0.76
EIF4E P06730 1/20 0.76
CYP3A4 P08684 1/20 0.76
TOP1 P11387 1/20 0.76
KDM4E B2RXH2 2/20 0.47
HTT P42858 2/20 0.47
BLM P54132 2/20 0.47
TP53 P04637 2/20 0.47
MAPT P10636 2/20 0.47
TDP1 Q9NUW8 1/20 0.47
GAA P10253 1/20 0.47
GMNN O75496 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Taribavirin SCHEMBL3868643 1.00 PNP (1.00) PNPLMNASMN1; SMN2ALDH1A1TSHR
Taribavirin SCHEMBL2619250 1.00 PNP (1.00) PNPLMNASMN1; SMN2ALDH1A1TSHR
Taribavirin SCHEMBL12758161 1.00 PNP (1.00) PNPLMNASMN1; SMN2ALDH1A1TSHR
Taribavirin SCHEMBL3307695 1.00 PNP (1.00) PNPLMNASMN1; SMN2ALDH1A1TSHR
Taribavirin SCHEMBL3307685 1.00 PNP (1.00) PNPLMNASMN1; SMN2ALDH1A1TSHR
Taribavirin SCHEMBL16330745 1.00 PNP (1.00) PNPLMNASMN1; SMN2ALDH1A1TSHR
Taribavirin SCHEMBL6981526 1.00 PNP (1.00) PNPLMNASMN1; SMN2ALDH1A1TSHR
Taribavirin SCHEMBL2631656 1.00 PNP (1.00) PNPLMNASMN1; SMN2ALDH1A1TSHR
Taribavirin SCHEMBL18735565 1.00 PNP (1.00) PNPLMNASMN1; SMN2ALDH1A1TSHR
Taribavirin SCHEMBL40670 1.00 PNP (1.00) PNPLMNASMN1; SMN2ALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3694512-A1 METHODS FOR TREATING HCV Abbvie Inc. (US) 2020-08-19 EP disclosed
WO-2019074507-A1 METHODS FOR TREATING HCV ABBVIE INC. (US) 2019-04-18 WO disclosed
WO-2017133517-A1 PHOSPHAMIDE DERIVATIVE, METHOD FOR MANUFACTURING THE SAME, AND USES THEREOF 四川海思科制药有限公司 2017-08-10 WO disclosed
EP-3125890-A1 METHODS FOR TREATING HCV AbbVie Inc. (US) 2017-02-08 EP disclosed
EP-3082808-A1 METHODS FOR TREATING LIVER TRANSPLANT RECIPIENTS AbbVie Inc. (US) 2016-10-26 EP disclosed
WO-2016134058-A1 COMBINATIONS USEFUL TO TREAT HEPATITIS C VIRUS ABBVIE INC. (US) 2016-08-25 WO disclosed
EP-2968302-A1 COMBINATION OF DIRECT ACTING ANTIVIRAL AGENTS AND RIBAVIRIN FOR TREATING HCV PATIENTS AbbVie Inc. (US) 2016-01-20 EP disclosed
WO-2015153792-A1 METHODS FOR TREATING HCV ABBVIE INC. (US) 2015-10-08 WO disclosed
WO-2015095572-A1 METHODS FOR TREATING LIVER TRANSPLANT RECIPIENTS ABBVIE INC. (US) 2015-06-25 WO disclosed
WO-2014152635-A9 COMBINATION OF DIRECT ACTING ANTIVIRAL AGENTS AND RIBAVIRIN FOR TREATING HCV PATIENTS ABBVIE INC. (US) 2014-12-11 WO disclosed
WO-2014152635-A1 COMBINATION OF DIRECT ACTING ANTIVIRAL AGENTS AND RIBAVIRIN FOR TREATING HCV PATIENTS ABBVIE INC. (US) 2014-09-25 WO disclosed
WO-2013059630-A1 METHODS FOR TREATING HCV COMPRISING AT LEAST TWO DIRECT ACTING ANTIVIRAL AGENT, RIBAVIRIN BUT NOT INTERFERON. ABBVIE INC. (US) 2013-04-25 WO disclosed
EP-1257281-B8 NUCLEOSIDE ANALOGS WITH CARBOXAMIDINE MODIFIED MONOCYCLIC BASE VALEANT PHARMACEUTICALS NORTH (US) 2008-01-23 EP disclosed
EP-1257281-A4 NUCLEOSIDE ANALOGS WITH CARBOXAMIDINE MODIFIED MONOCYCLIC BASE ICN PHARMACEUTICALS (US) 2003-03-19 EP disclosed
EP-1257281-A1 NUCLEOSIDE ANALOGS WITH CARBOXAMIDINE MODIFIED MONOCYCLIC BASE ICN Pharmaceuticals, Inc. (US) 2002-11-20 EP disclosed
WO-2001060379-A1 NUCLEOSIDE ANALOGS WITH CARBOXAMIDINE MODIFIED MONOCYCLIC BASE RIBAPHARM CORP. (US) 2001-08-23 WO disclosed