SCHEMBL263167

SCHEMBL263167

CCOP(=O)(OCC)C(F)(F)Br

nearest known ligand 0.43

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.43
TP53 P04637 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
PPARD Q03181 2/20 0.34
NPSR1 Q6W5P4 1/20 0.33
KCNH2 Q12809 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19772489 0.89 MEN1 (0.36) TSHRTP53TDP1
SCHEMBL25463304 0.89 TSHR (0.39) TSHRTP53TDP1PPARDNPSR1
SCHEMBL4757795 0.85 TSHR (0.43) TSHRTP53TDP1PPARDNPSR1
SCHEMBL3146731 0.79 TSHR (0.48) TSHRTP53TDP1PPARDNPSR1
SCHEMBL9614639 0.79 TSHR (0.48) TSHRTP53TDP1PPARDNPSR1
SCHEMBL10426582 0.79 TSHR (0.48) TSHRTP53TDP1PPARD
SCHEMBL4434268 0.79 TSHR (0.48) TSHRTP53TDP1PPARD
SCHEMBL18087213 0.78 TSHR (0.42) TSHRTP53TDP1PPARDNPSR1
SCHEMBL10128271 0.77 TSHR (0.46) TSHRTP53TDP1PPARD
SCHEMBL3502263 0.76 TSHR (0.40) TSHRTP53TDP1PPARD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1032 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-122036711-A Pyricularia sulfone Synthesis method of intermediate 山东潍坊润丰化工股份有限公司 2026-05-15 CN claimed
CN-114085234-B Process for preparing 1, 3-benzodioxole heterocyclic compounds 联合疗法公司 2024-12-17 CN claimed
EP-3390407-B1 METHODS FOR THE PREPARATION OF 1,3-BENZODIOXOLE HETEROCYCLIC COMPOUNDS UNION THERAPEUTICS AS (DK) 2023-10-11 EP claimed
US-11760701-B2 Difluoromethoxylation and trifluoromethoxylation compositions and methods for synthesizing same THE RESEARCH FOUNDATION FOR THE STATE UNIVERSITY OF NEW YROK (US) 2023-09-19 US claimed
US-20230073362-A1 METHODS FOR THE PREPARATION OF 1,3-BENZODIOXOLE HETEROCYCLIC COMPOUNDS UNION therapeutics A/S (DK) 2023-03-09 US claimed
US-11370799-B2 Methods for the preparation of 1,3-benzodioxole heterocyclic compounds UNION therapeutics A/S (DK) 2022-06-28 US claimed
US-20220162227-A1 METHODS FOR THE PREPARATION OF 1,3-BENZODIOXOLE HETEROCYCLIC COMPOUNDS UNION therapeutics A/S (DK) 2022-05-26 US claimed
US-20200262842-A1 METHODS FOR THE PREPARATION OF 1,3-BENZODIOXOLE HETEROCYCLIC COMPOUNDS UNION therapeutics A/S (DK) 2020-08-20 US claimed
US-12637435-B2 Nitrogen-containing heterocyclic compound or salt thereof, use thereof, and intermediate thereof FUJIFILM CORPORATION (JP) 2026-05-26 US disclosed
CN-122074043-A Combination therapy with KRAS modulators 光达治疗公司 2026-05-22 CN disclosed
WO-2026107227-A1 COMPOSITIONS COMPRISING USP1 INHIBITORS AND METHODS OF USING THE SAME EIKON THERAPEUTICS, INC. (US) 2026-05-21 WO disclosed
US-20260138977-A1 MODULATORS OF BETA CATENIN AND USES THEREOF DEWPOINT THERAPEUTICS INC (US) 2026-05-21 US disclosed
EP-4744661-A2 NOVEL PYRIMIDIN-2-YL SULFONAMIDE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2026-05-20 EP disclosed
US-12630514-B2 Process and intermediates for the preparation of pyroxasulfone ADAMA AGAN LTD. (IL) 2026-05-19 US disclosed
US-5538978-A NUCLEOSIDE PHOSPHORYLASE INHIBITORS AS IMMUNOSUPPRESSANTS, ANTILYMPHOMA, ANTILEUKEMIA, VIRICIDES AND ANTIPROTOZOA AGENTS MERRELL PHARMACEUTICALS INC. (US) 1996-07-23 US disclosed
US-5527803-A IMMUNOSUPPRESSANTS, PHOSPHORYLASE INHIBITORS MERRELL PHARMACEUTICALS INC. (US) 1996-06-18 US disclosed
US-5494912-A 9-purinyl phosphonic acid derivitives for treating gout MERRELL PHARMACEUTICALS INC. (US) 1996-02-27 US disclosed
EP-0465297-B1 9-Purinyl phosphonic acid derivatives MERRELL DOW PHARMA (US) 1996-01-31 EP disclosed
EP-0531597-A1 Novel unsaturated acyclic phosphonate derivatives of purine and pyrimidine MERRELL DOW PHARMACEUTICALS INC. (US) 1993-03-17 EP disclosed
EP-0465297-A1 9-Purinyl phosphonic acid derivatives MERRELL PHARMACEUTICALS INC. (US) 1992-01-08 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200262842-A1 METHODS FOR THE PREPARATION OF 1,3-BENZODIOXOLE HETEROCYCLIC COMPOUNDS PDE4B, PDE4A, PDE4C TSHR 3441/4885TP53 4715/4885TDP1 203/4885
US-20230073362-A1 METHODS FOR THE PREPARATION OF 1,3-BENZODIOXOLE HETEROCYCLIC COMPOUNDS PDE4B, PDE4A, PDE3B TSHR 3679/4885TP53 4701/4885TDP1 183/4885
US-12630514-B2 Process and intermediates for the preparation of pyroxasulfone MRPS23, CYP2E1, CYP2S1 TSHR 1582/4885TP53 2598/4885TDP1 2101/4885
US-20260138977-A1 MODULATORS OF BETA CATENIN AND USES THEREOF CTNNB1, CTNND1, CTNNA1 TSHR 4681/4885TP53 61/4885TDP1 861/4885
US-12637435-B2 Nitrogen-containing heterocyclic compound or salt thereof, use thereof, and intermediate thereof CBR1, DHODH, CBR3 TSHR 2492/4885TP53 686/4885TDP1 2604/4885
US-11760701-B2 Difluoromethoxylation and trifluoromethoxylation compositions and methods for synthesizing same AFF2, AFF4, AFF1 TSHR 2337/4885TP53 1099/4885TDP1 2207/4885
US-20220162227-A1 METHODS FOR THE PREPARATION OF 1,3-BENZODIOXOLE HETEROCYCLIC COMPOUNDS PDE4B, PDE4A, PDE4C TSHR 3696/4885TP53 4732/4885TDP1 185/4885
US-11370799-B2 Methods for the preparation of 1,3-benzodioxole heterocyclic compounds PDE4B, PDE4A, PDE4C TSHR 3441/4885TP53 4715/4885TDP1 203/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.