Eflornithine

Eflornithine

SCHEMBL26327

NCCCC(N)(C(=O)O)C(F)F

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ODC1

The experimentally established mechanism targets of Eflornithine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ODC1 known ✓ P11926 2/20 1.00
LMNA P02545 3/20 0.96
BLM P54132 3/20 0.96
KDM4E B2RXH2 1/20 0.96
MAPT P10636 1/20 0.96
RAB9A P51151 1/20 0.96
PMP22 Q01453 1/20 0.96
SMN1; SMN2 Q16637 1/20 0.96
ARG1 P05089 3/20 0.62
ARG2 P78540 2/20 0.41
THRB P10828 2/20 0.34
KMT2A Q03164 2/20 0.34
NPSR1 Q6W5P4 2/20 0.34
GABRR3 A8MPY1 1/20 0.34
GABRP O00591 1/20 0.34
GABRD O14764 1/20 0.34
HDAC3 O15379 1/20 0.34
GABBR2 O75899 1/20 0.34
CYP1A2 P05177 1/20 0.34
GABRA1 P14867 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Eflornithine, (S)- SCHEMBL60698 1.00 ODC1 (1.00) ODC1LMNABLMKDM4EMAPT
D-Eflornithine SCHEMBL60699 1.00 ODC1 (1.00) ODC1LMNABLMKDM4EMAPT
Eflornithine SCHEMBL8581344 1.00 ODC1 (1.00) ODC1LMNABLMKDM4EMAPT
D-Eflornithine SCHEMBL7208883 0.98 BLM (1.00) ODC1LMNABLMKDM4EMAPT
Eflornithine SCHEMBL6779168 0.98 BLM (1.00) ODC1LMNABLMKDM4EMAPT
Eflornithine SCHEMBL3244711 0.98 ODC1 (0.96) ODC1LMNABLMKDM4EMAPT
Eflornithine, (S)- SCHEMBL6779172 0.98 BLM (1.00) ODC1LMNABLMKDM4EMAPT
Eflornithine SCHEMBL3022583 0.98 BLM (1.00) ODC1LMNABLMKDM4EMAPT
Eflornithine, (S)- SCHEMBL1322403 0.98 BLM (1.00) ODC1LMNABLMKDM4EMAPT
D-Eflornithine SCHEMBL3244719 0.98 ODC1 (0.96) ODC1LMNABLMKDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 29032 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4748859-A2 CHEMICALLY AND PHOTOCHEMICALLY INITIATED CELL MEMBRANE BLEBBING TO INDUCE CELL VESICLE PRODUCTION, MODIFICATIONS THEREOF, AND USES THEREOF The Regents of the University of California (US) 2026-05-27 EP claimed
EP-3368029-B1 EFLORNITHINE AND SULINDAC, FIXED DOSE COMBINATION FORMULATION USWM LLC (US) 2026-05-27 EP claimed
US-20260137642-A1 METHODS OF TREATING PATIENTS HAVING TYPE 1 DIABETES WITH EFLORNITHINE CANCER PREVENTION PHARMACEUTICALS, INC. (US) 2026-05-21 US claimed
US-20260137794-A1 LIGAND-DRUG CONJUGATE AND USE THEREOF SYSTIMMUNE INC (US) 2026-05-21 US claimed
EP-4743490-A1 HUMANIZED ANTI-CD7 ANTIBODY Christian-Albrechts-Universität zu Kiel (DE) 2026-05-20 EP claimed
WO-2026099502-A1 NOVEL DRUG CONJUGATES FOR TESTING CELLULAR DRUG UPTAKE Deutsches Krebsforschungszentrum Stiftung des öffentlichen Rechts (DE) 2026-05-15 WO claimed
EP-4255391-B1 LUMINOL FOR USE IN THE TREATMENT OF SEQUELAE OF A SARS-COV-2 INFECTION METRIOPHARM AG (CH) 2026-05-06 EP claimed
US-20260116861-A1 ISOXAZOLE HYDROXAMIC ACIDS AS HISTONE DEACETYLASE 6 INHIBITORS THE GEORGE WASHINGTON UNIVERSITY, A CONGRESSIONALLY CHARTERED NOT-FOR-PROFIT CORPORATION (US) 2026-04-30 US claimed
US-20260108451-A1 COMPOSITIONS FOR THE MANAGEMENT OF HIRSUTISM MAJEED ANJU (IN) 2026-04-23 US claimed
US-20260108619-A1 CONJUGATION LINKERS, CELL BINDING MOLECULE-DRUG CONJUGATES CONTAINING THE LINKERS, METHODS OF MAKING AND USES SUCH CONJUGATES WITH THE LINKERS HANGZHOU DAC BIOTECH CO., LTD. (CN) 2026-04-23 US claimed
EP-0211354-A2 Nucleosides and their use as antineoplastic agents MERRELL DOW PHARMACEUTICALS INC. (US) 1987-02-25 EP claimed
EP-0198893-A1 HAIR GROWTH MODIFICATION. HANDELMAN JOSEPH H (US) 1986-10-29 EP claimed
WO-1986002269-A1 HAIR GROWTH MODIFICATION HANDELMAN, JOSEPH, H. (US) 1986-04-24 WO claimed
EP-0162413-A2 Polyamine for use as a medicine in the treatment of neoplasms MERRELL DOW PHARMACEUTICALS INC. (US) 1985-11-27 EP claimed
US-4499072-A Process for treating diseases with ODC inhibitors MERRELL DOW PHARMACEUTICALS INC. (US) 1985-02-12 US claimed
US-4496588-A HALOMETHYL DERIVATIVES OF A-AMINO ACID MERRELL TORAUDE ET COMPAGNIE (FR) 1985-01-29 US claimed
US-4433051-A Derivatives of α-difluoromethylornithine useful in analysis YEDA RESEARCH AND DEVELOPMENT CO., LTD. (IS) 1984-02-21 US claimed
US-4413141-A INHIBITOR OF ORNITHINE DECARBOXYLASE MERRELL TORAUDE ET COMPAGNIE (FR) 1983-11-01 US claimed
US-4336054-A AMINO ACIDS MERRELL DOW PHARMACEUTICALS INC. (US) 1982-06-22 US claimed
US-4330559-A 2,5-DIAMINO-2-FLUOROMETHYLPENTANOIC ACIDS OR DERIVATIVES MERRELL-TORAUDE ET CIE (FR) 1982-05-18 US claimed