SCHEMBL2632824

SCHEMBL2632824

CCn1c(=O)c(-c2ccc(OC)cc2OC)cc2c(C)nc(NCCF)nc21

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.46
ALDH1A1 P00352 1/20 0.46
GLA P06280 1/20 0.46
GAA P10253 1/20 0.46
HPGD P15428 1/20 0.46
MAPK1 P28482 1/20 0.46
HTT P42858 1/20 0.46
HSD17B10 Q99714 1/20 0.46
RXFP1 Q9HBX9 1/20 0.46
CRHR1 P34998 6/20 0.45
PIK3CA P42336 10/20 0.43
PIK3CD O00329 1/20 0.38
PIK3CB P42338 1/20 0.38
MTOR P42345 1/20 0.38
PIK3CG P48736 1/20 0.38
BCDIN3D Q7Z5W3 1/20 0.38
ADORA3 P0DMS8 1/20 0.37
FGFR1 P11362 1/20 0.36
FGFR2 P21802 1/20 0.36
FGFR4 P22455 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL188683 0.91 ALDH1A1 (0.57) KDM4EALDH1A1GLAGAAHPGD
SCHEMBL189196 0.79 HSD17B10 (0.59) KDM4EALDH1A1GLAGAAHPGD
SCHEMBL189483 0.77 ALDH1A1 (0.60) KDM4EALDH1A1GLAGAAHPGD
SCHEMBL14548188 0.77 ALDH1A1 (0.53) KDM4EALDH1A1GLAGAAHPGD
SCHEMBL189211 0.76 PIK3CA (0.67) KDM4EALDH1A1GLAGAAHPGD
SCHEMBL188808 0.75 PIK3CA (0.71) KDM4EALDH1A1GLAGAAHPGD
SCHEMBL188692 0.71 ALDH1A1 (0.60) KDM4EALDH1A1GLAGAAHPGD
SCHEMBL188697 0.70 ALDH1A1 (0.61) KDM4EALDH1A1GLAGAAHPGD
SCHEMBL190012 0.69 KDM4E (0.60) KDM4EALDH1A1GLAGAAHPGD
SCHEMBL189082 0.69 ALDH1A1 (0.57) KDM4EALDH1A1GLAGAAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2056829-B9 USING PI3K AND MEK MODULATORS IN TREATMENTS OF CANCER EXELIXIS INC (US) 2012-09-26 EP disclosed