SCHEMBL26330322

SCHEMBL26330322

Cc1nc2c3cccc(Cl)c3nc(N)n2n1

nearest known ligand 0.52

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HSP90AB1 P08238 2/20 0.52
ADORA2A P29274 9/20 0.50
NR4A2 P43354 1/20 0.48
PARP1 P09874 1/20 0.43
PDE10A Q9Y233 3/20 0.40
HAVCR2 Q8TDQ0 3/20 0.40
HSD17B10 Q99714 1/20 0.40
ACHE P22303 1/20 0.38
ADORA2B P29275 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17897308 0.80 ADORA2A (0.57) HSP90AB1ADORA2A
SCHEMBL15846590 0.77 ADORA2A (0.46) HSP90AB1ADORA2APDE10AHAVCR2HSD17B10
SCHEMBL14810416 0.76 ADORA2A (0.67) ADORA2AADORA2B
SCHEMBL19104709 0.76 HSP90AB1 (0.46) HSP90AB1ADORA2ANR4A2
SCHEMBL18948427 0.75 PDE10A (0.63) HSP90AB1PDE10AHAVCR2HSD17B10
SCHEMBL22987876 0.75 ADORA2A (0.48) HSP90AB1ADORA2AADORA2B
SCHEMBL22987894 0.74 HSP90AB1 (0.45) HSP90AB1ADORA2ANR4A2ADORA2B
SCHEMBL19941816 0.71 HSP90AB1 (0.44) HSP90AB1ADORA2A
SCHEMBL26330327 0.69 ADORA2A (0.48) ADORA2APDE10AADORA2B
SCHEMBL15846588 0.66 HSP90AB1 (0.45) HSP90AB1ADORA2AHSD17B10ADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023158626-A1 ADENOSINE RECEPTOR ANTAGONISTS, PHARMACEUTICAL COMPOSITIONS AND THEIR USE THEREOF MERCK SHARP & DOHME LLC (US) 2023-08-24 WO disclosed