SCHEMBL2635560

SCHEMBL2635560

CCOC(=O)N(c1c(C)noc1-c1ccc(-c2ccc(C3(C(=O)OCC)CC3)cc2)cc1)C1CC1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ABCC3 O15438 1/20 0.41
ABCC4 O15439 1/20 0.41
ABCB11 O95342 1/20 0.41
CYP2C8 P10632 1/20 0.41
CYP2C9 P11712 1/20 0.41
ABCB4 P21439 1/20 0.41
LPAR1 Q92633 1/20 0.41
ABCC2 Q92887 1/20 0.41
SLCO1B3 Q9NPD5 1/20 0.41
SLCO1B1 Q9Y6L6 1/20 0.41
OPRM1 P35372 9/20 0.39
OPRD1 P41143 3/20 0.37
OPRK1 P41145 3/20 0.37
SLC22A1 O15245 1/20 0.37
SLC6A4 P31645 1/20 0.37
ADRA1A P35348 1/20 0.37
KCNH2 Q12809 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2636805 0.97 SLCO1B1 (0.38) ABCC3ABCC4ABCB11CYP2C8CYP2C9
SCHEMBL2635538 0.95 SLC6A9 (0.40) ABCC3ABCC4ABCB11CYP2C8CYP2C9
SCHEMBL2635693 0.93 LPAR1 (0.48) ABCC3ABCC4ABCB11CYP2C8CYP2C9
SCHEMBL2635736 0.90 LPAR1 (0.45) ABCC3ABCC4ABCB11CYP2C8CYP2C9
SCHEMBL2761762 0.89 SLCO1B1 (0.34) ABCC3ABCC4ABCB11CYP2C8CYP2C9
SCHEMBL2636376 0.89 LPAR1 (0.44) ABCC3ABCC4ABCB11CYP2C8CYP2C9
SCHEMBL2761409 0.87 SLCO1B1 (0.33) ABCC3ABCC4ABCB11CYP2C8CYP2C9
SCHEMBL2761822 0.85 SLCO1B1 (0.36) ABCC3ABCC4ABCB11CYP2C8CYP2C9
SCHEMBL6894 0.82 SLC6A9 (0.41) ABCC3ABCC4ABCB11CYP2C8CYP2C9
SCHEMBL2761346 0.82 CA12 (0.40) LPAR1SLCO1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2438048-A2 POLYCYCLIC ANTAGONISTS OF LYSOPHOSPHATIDIC ACID RECEPTORS Amira Pharmaceuticals, Inc. (US) 2012-04-11 EP disclosed
WO-2010141768-A2 POLYCYCLIC ANTAGONISTS OF LYSOPHOSPHATIDIC ACID RECEPTORS AMIRA PHARMACEUTICALS, INC. (US) 2010-12-09 WO disclosed
WO-2010141761-A2 POLYCYCLIC ANTAGONISTS OF LYSOPHOSPHATIDIC ACID RECEPTORS AMIRA PHARMACEUTICALS, INC. (US) 2010-12-09 WO disclosed