SCHEMBL26358255

SCHEMBL26358255

CC(C)Oc1ccn2c(-c3cncc(N[C@H]4CCCC[C@@H]4F)n3)cnc2c1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
FLT3 P36888 7/20 0.43
KDR P35968 7/20 0.34
CSF1R P07333 6/20 0.34
KIT P10721 5/20 0.34
CYP2D6 P10635 1/20 0.34
KCNH2 Q12809 1/20 0.34
DYRK1A Q13627 4/20 0.33
CLK2 P49760 2/20 0.33
CLK3 P49761 2/20 0.33
GSK3B P49841 2/20 0.33
IGF1R P08069 1/20 0.33
IRAK4 Q9NWZ3 1/20 0.33
PIM1 P11309 1/20 0.33
PIM3 Q86V86 1/20 0.33
PIM2 Q9P1W9 1/20 0.33
ABL1 P00519 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26358257 0.98 FLT3 (0.43) FLT3KDRCSF1RKITCYP2D6
SCHEMBL26358046 0.89 FLT3 (0.54) FLT3KDRCSF1RKITCYP2D6
SCHEMBL24232004 0.89 FLT3 (0.47) FLT3KDRCSF1RKITCYP2D6
SCHEMBL26358053 0.88 FLT3 (0.41) FLT3KDRCSF1RKITCYP2D6
SCHEMBL24231493 0.87 FLT3 (0.52) FLT3KDRCSF1RKITCYP2D6
SCHEMBL26357442 0.87 FLT3 (0.54) FLT3KDRCSF1RKITCYP2D6
SCHEMBL26358260 0.85 MAPK8 (0.42) FLT3KDRCSF1RKITCYP2D6
SCHEMBL26358267 0.85 FLT3 (0.39) FLT3KDRCSF1RKITCYP2D6
SCHEMBL26358253 0.83 FLT3 (0.39) FLT3KDRCSF1RKITCYP2D6
SCHEMBL26358263 0.83 MAPK8 (0.42) FLT3KDRCSF1RKITCYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230303563-A1 MULTI-CYCLIC IRAK AND FLT3 INHIBITING COMPOUNDS AND USES THEREOF CHILDREN'S HOSPITAL MEDICAL CENTER 2023-09-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230303563-A1 MULTI-CYCLIC IRAK AND FLT3 INHIBITING COMPOUNDS AND USES THEREOF FLT3, IRAK2, IRAK3 FLT3 1/4885KDR 640/4885CSF1R 40/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.