SCHEMBL26358053

SCHEMBL26358053

CC(C)Oc1ccn2c(-c3cc(F)cc(N[C@H]4CCCC[C@@H]4F)n3)cnc2c1

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
FLT3 P36888 9/20 0.41
KDR P35968 9/20 0.34
CSF1R P07333 6/20 0.34
KIT P10721 3/20 0.34
CYP2D6 P10635 1/20 0.34
KCNH2 Q12809 1/20 0.34
IRAK4 Q9NWZ3 2/20 0.33
ALOX5AP P20292 1/20 0.32
FEN1 P39748 1/20 0.32
ABL1 P00519 1/20 0.32
SIK1 P57059 1/20 0.31
SIK2 Q9H0K1 1/20 0.31
SIK3 Q9Y2K2 1/20 0.31
IGF1R P08069 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24231379 0.89 FLT3 (0.45) FLT3KDRCSF1RKITCYP2D6
SCHEMBL25991407 0.89 FLT3 (0.45) FLT3KDRCSF1RKITCYP2D6
SCHEMBL26358255 0.88 FLT3 (0.43) FLT3KDRCSF1RKITCYP2D6
SCHEMBL26358046 0.88 FLT3 (0.54) FLT3KDRCSF1RKITCYP2D6
SCHEMBL24231319 0.88 FLT3 (0.49) FLT3KDRCSF1RKITCYP2D6
SCHEMBL25989698 0.88 FLT3 (0.49) FLT3KDRCSF1RKITCYP2D6
SCHEMBL26358257 0.86 FLT3 (0.43) FLT3KDRCSF1RKITCYP2D6
SCHEMBL26357442 0.86 FLT3 (0.54) FLT3KDRCSF1RKITCYP2D6
SCHEMBL26358267 0.84 FLT3 (0.39) FLT3KDRCSF1RKITCYP2D6
SCHEMBL26358260 0.84 MAPK8 (0.42) FLT3KDRCSF1RKITCYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230303563-A1 MULTI-CYCLIC IRAK AND FLT3 INHIBITING COMPOUNDS AND USES THEREOF CHILDREN'S HOSPITAL MEDICAL CENTER 2023-09-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230303563-A1 MULTI-CYCLIC IRAK AND FLT3 INHIBITING COMPOUNDS AND USES THEREOF FLT3, IRAK2, IRAK3 FLT3 1/4885KDR 640/4885CSF1R 40/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.