SCHEMBL263592

SCHEMBL263592

NCc1ccc2[nH]nnc2c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.42
PKM P14618 1/20 0.42
LOXL2 Q9Y4K0 5/20 0.33
HRH3 Q9Y5N1 1/20 0.33
LOX P28300 1/20 0.33
LOXL3 P58215 1/20 0.33
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA3 P07451 1/20 0.33
CA4 P22748 1/20 0.33
CA6 P23280 1/20 0.33
CA5A P35218 1/20 0.33
CA7 P43166 1/20 0.33
CA9 Q16790 1/20 0.33
CA14 Q9ULX7 1/20 0.33
CA5B Q9Y2D0 1/20 0.33
ROCK1 Q13464 1/20 0.33
AKT2 P31751 1/20 0.32
CYP2A6 P11509 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7214713 0.98 GAA (0.44) GAAPKMLOXL2HRH3LOX
SCHEMBL12686295 0.85 GAA (0.42) GAAPKMLOXL2HRH3LOX
SCHEMBL501616 0.84 MEN1 (0.39) CA1CA2CA4CA6
SCHEMBL7127295 0.81
SCHEMBL241363 0.81 TP53 (0.37) GAACA12CA9CYP2A6NOS1
SCHEMBL3824241 0.81
SCHEMBL31262817 0.81 HSD17B10 (0.39) CA12CA2CA3CA4CA6
SCHEMBL1692572 0.81 HSD17B10 (0.39) CA12CA2CA3CA4CA6
SCHEMBL5016026 0.80 IDO1 (0.42)
SCHEMBL6364875 0.79 TP53 (0.36) GAACA12CA9CYP2A6NOS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112778274-B Nitrogen-containing heterocyclic derivative and preparation thereof 四川海思科制药有限公司 2022-02-15 CN disclosed
WO-2021214472-A1 TETRAHYDROISOQUINOLINE COMPOUNDS AS NRF2 ACTIVATORS C4X DISCOVERY LIMITED (GB) 2021-10-28 WO disclosed
US-20180194751-A1 INDOLE DERIVATIVE, PREPARATION METHOD THEREOF, AND USE THEREOF IN PHARMACEUTICAL DRUG ZHEJIANG HISUN PHARMACEUTICAL CO., LTD. (CN) 2018-07-12 US disclosed
US-8134004-B2 Substituted N-bicyclicalkyl bicycliccarboxyamide compounds PFIZER INC. (US) 2012-03-13 US disclosed
US-20090253740-A1 SUBSTITUTED N-BICYCLICALKYL BICYCLICCARBOXYAMIDE COMPOUNDS PFIZER INC 2009-10-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090253740-A1 SUBSTITUTED N-BICYCLICALKYL BICYCLICCARBOXYAMIDE COMPOUNDS OPRL1, CNR1, TRPV1 GAA 2833/4885PKM 2147/4885LOXL2 2596/4885
US-20180194751-A1 INDOLE DERIVATIVE, PREPARATION METHOD THEREOF, AND USE THEREOF IN PHARMACEUTICAL DRUG FGFR1, FGFR2, FGFR4 GAA 3574/4885PKM 2821/4885LOXL2 2876/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.