SCHEMBL2635931

SCHEMBL2635931

CCCCOC(=O)OC(=O)Nc1ncc(-c2ccc(=O)[nH]c2C(C)C)nc1-c1cc(-c2cccc(CCl)c2)no1

nearest known ligand 0.35

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ATR Q13535 4/20 0.35
PPARG P37231 2/20 0.34
PPARA Q07869 2/20 0.34
AGTR2 P50052 3/20 0.31
PTPN1 P18031 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2B6 P20813 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2635929 0.83 PPARG (0.35) ATRPPARGPPARAPTPN1
SCHEMBL2635934 0.66 ATR (0.53) ATRPPARGPPARA
SCHEMBL2635709 0.64 ATR (0.55) ATR
SCHEMBL2637131 0.62 ATM (0.39) ATRPTPN1
SCHEMBL506418 0.59 ATR (0.81) ATR
SCHEMBL2635705 0.58 ATR (0.51) ATR
SCHEMBL2635675 0.57 ATR (0.38) ATRPPARA
SCHEMBL2635523 0.57 ATR (0.69) ATR
SCHEMBL22502725 0.57 RAB9A (0.44) CYP2C9
SCHEMBL2634728 0.56 ATR (0.39) ATR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2569313-A1 COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE Vertex Pharmaceuticals Incorporated (US) 2013-03-20 EP disclosed
WO-2011143426-A1 COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE VERTEX PHARMACEUTICALS INCORPORATED (US) 2011-11-17 WO disclosed