SCHEMBL2637564

SCHEMBL2637564

COCCOc1ccc2cncnc2c1

nearest known ligand 0.69

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
EGFR P00533 7/20 0.69
KDM1A O60341 1/20 0.42
PDGFRB P09619 1/20 0.42
PDGFRA P16234 1/20 0.42
NCF1 P14598 4/20 0.42
ILK Q13418 1/20 0.41
FGFR1 P11362 1/20 0.41
FLT1 P17948 1/20 0.41
KDR P35968 1/20 0.41
HPGDS O60760 2/20 0.41
APP P05067 1/20 0.40
FBP1 P09467 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
HDAC5 Q9UQL6 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7140894 0.96 EGFR (0.63) EGFRKDM1ANCF1ILKAPP
SCHEMBL29831918 0.84 EGFR (0.59) EGFRNCF1
SCHEMBL30504578 0.82 EGFR (0.70) EGFRPDGFRBPDGFRANCF1HDAC1
SCHEMBL4649110 0.82 EGFR (0.70) EGFRPDGFRBPDGFRANCF1HDAC1
SCHEMBL30241125 0.82 EGFR (1.00) EGFRPDGFRBPDGFRAHPGDS
SCHEMBL668493 0.82 EGFR (1.00) EGFRPDGFRBPDGFRAHPGDS
SCHEMBL29517021 0.82 EGFR (1.00) EGFRPDGFRBPDGFRAHPGDS
SCHEMBL6489451 0.81 EGFR (0.59) EGFRPDGFRBPDGFRANCF1HDAC1
Hydrochloric Acid SCHEMBL28023744 0.80 EGFR (0.96) EGFRPDGFRBPDGFRAHPGDS
SCHEMBL5682759 0.79 EGFR (0.56) EGFRNCF1HDAC1HDAC6HDAC5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3436446-B1 MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR VERTEX PHARMA (US) 2023-06-07 EP disclosed
EP-2569298-A1 NOVEL CCR2 RECEPTOR ANTAGONISTS, METHOD FOR PRODUCING THE SAME, AND USE THEREOF AS MEDICAMENTS Boehringer Ingelheim International GmbH (DE) 2013-03-20 EP disclosed
WO-2011141474-A1 NOVEL CCR2 RECEPTOR ANTAGONISTS, METHOD FOR PRODUCING THE SAME, AND USE THEREOF AS MEDICAMENTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-11-17 WO disclosed
EP-1799191-A1 MODIFYING SURFACES OF LACTOSE SERVING AS AN AUXILIARY AGENT TO BE USED FOR POWDER INHALANTS Boehringer Ingelheim International GmbH (DE) 2007-06-27 EP disclosed
WO-2006037738-A1 MODIFYING SURFACES OF LACTOSE SERVING AS AN AUXILIARY AGENT TO BE USED FOR POWDER INHALANTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2006-04-13 WO disclosed