SCHEMBL2637798

SCHEMBL2637798

O=c1cc2[nH]c(-c3cccc(C(F)(F)F)c3)cc(=O)n2[nH]1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SCN2A Q99250 3/20 0.44
LDHA P00338 1/20 0.43
MAPT P10636 1/20 0.43
XDH P47989 1/20 0.43
TYMP P19971 1/20 0.43
CDC7 O00311 1/20 0.40
MAP4K4 O95819 1/20 0.39
PIM1 P11309 1/20 0.39
GPX4 P36969 1/20 0.39
GSK3B P49841 1/20 0.39
PIM3 Q86V86 1/20 0.39
BRSK1 Q8TDC3 1/20 0.39
MAP4K5 Q9Y4K4 1/20 0.39
NOTUM Q6P988 1/20 0.39
NPY5R Q15761 1/20 0.39
MAPK14 Q16539 1/20 0.39
KDM5B Q9UGL1 1/20 0.38
HTT P42858 1/20 0.37
ALKBH5 Q6P6C2 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2637446 0.85 RAD51 (0.43) SCN2ATYMPGSK3B
SCHEMBL12952973 0.76 SCN2A (0.47) SCN2ALDHAMAPTXDHTYMP
SCHEMBL10275874 0.69 MAPT (0.42) SCN2AMAPTMAPK14
SCHEMBL9376640 0.68 MAPT (0.40) SCN2ALDHAMAPTNPY5RHTT
SCHEMBL2490895 0.66 BRD4 (0.60) SCN2ALDHAMAPTXDHCDC7
SCHEMBL29678302 0.65 TSHR (0.58) SCN2ANOTUM
SCHEMBL1263144 0.65 TSHR (0.58) SCN2ANOTUM
SCHEMBL4305000 0.64 TNKS (0.44) SCN2AMAPTXDHNOTUMNPY5R
Ammonia Solution, Strong SCHEMBL20472961 0.63 MAOB (0.56) SCN2ANOTUM
SCHEMBL12049289 0.63 KDM4E (0.45) SCN2AMAPTMAPK14HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2438070-A1 GLYCINE B ANTAGONISTS Merz Pharma GmbH & Co. KGaA (DE) 2012-04-11 EP claimed
WO-2010139483-A1 GLYCINE B ANTAGONISTS MERZ PHARMA GMBH & CO. KGAA (DE) 2010-12-09 WO claimed
EP-2438070-A1 GLYCINE B ANTAGONISTS Merz Pharma GmbH & Co. KGaA (DE) 2012-04-11 EP disclosed
WO-2010139483-A1 GLYCINE B ANTAGONISTS MERZ PHARMA GMBH & CO. KGAA (DE) 2010-12-09 WO disclosed