SCHEMBL2637446

SCHEMBL2637446

O=c1cc2[nH]c(-c3ccc(C(F)(F)F)cc3)cc(=O)n2[nH]1

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
RAD51 Q06609 3/20 0.43
PARP1 P09874 1/20 0.42
TNKS O95271 1/20 0.42
CCNB2 O95067 1/20 0.40
CDK1 P06493 1/20 0.40
CCNB1 P14635 1/20 0.40
GSK3A P49840 1/20 0.40
GSK3B P49841 1/20 0.40
CCNB3 Q8WWL7 1/20 0.40
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
TYMP P19971 1/20 0.38
HDAC11 Q96DB2 2/20 0.36
GLO1 Q04760 1/20 0.35
RAB9A P51151 1/20 0.35
SCN2A Q99250 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2637798 0.85 SCN2A (0.44) GSK3BTYMPSCN2A
SCHEMBL10282683 0.83 RAD51 (0.44) RAD51PARP1TNKSCCNB2CDK1
SCHEMBL10275874 0.77 MAPT (0.42) PARP1TNKSKDM4EALDH1A1LMNA
SCHEMBL2087491 0.72 PARP1 (0.50) PARP1TNKSCCNB2CDK1CCNB1
SCHEMBL3561170 0.68 PARP1 (0.47) PARP1TNKSCCNB2CDK1CCNB1
SCHEMBL19073622 0.67 TNKS (0.43) PARP1TNKSCCNB2CDK1CCNB1
SCHEMBL8987300 0.66 KIF11 (0.56) PARP1TNKSCCNB2CDK1CCNB1
SCHEMBL8987203 0.66 KIF11 (0.56) PARP1TNKSCCNB2CDK1CCNB1
SCHEMBL3558874 0.65 KDM4E (0.50) PARP1TNKSCCNB2CDK1CCNB1
SCHEMBL10275822 0.65 ALDH1A1 (0.68) TNKSKDM4EALDH1A1LMNARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2438070-A1 GLYCINE B ANTAGONISTS Merz Pharma GmbH & Co. KGaA (DE) 2012-04-11 EP claimed
WO-2010139483-A1 GLYCINE B ANTAGONISTS MERZ PHARMA GMBH & CO. KGAA (DE) 2010-12-09 WO claimed
EP-2438070-A1 GLYCINE B ANTAGONISTS Merz Pharma GmbH & Co. KGaA (DE) 2012-04-11 EP disclosed
WO-2010139483-A1 GLYCINE B ANTAGONISTS MERZ PHARMA GMBH & CO. KGAA (DE) 2010-12-09 WO disclosed