SCHEMBL2637833

SCHEMBL2637833

Cc1nc(C(C)C)c(-c2ccnc(Nc3ncc(C(=O)Nc4cc(-c5ccc(F)cc5)ccc4N)s3)n2)[nH]1

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HDAC2 Q92769 14/20 0.46
HDAC3 O15379 10/20 0.46
HDAC1 Q13547 6/20 0.39
KCNH2 Q12809 2/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2C18 P33260 1/20 0.39
CYP2C19 P33261 1/20 0.39
ABL1 P00519 2/20 0.37
BCR P11274 1/20 0.37
GSK3B P49841 1/20 0.36
MAPK14 Q16539 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2638901 0.89 HDAC2 (0.43) HDAC2HDAC3HDAC1KCNH2CYP1A2
SCHEMBL2637841 0.89 HDAC2 (0.43) HDAC2HDAC3HDAC1KCNH2CYP1A2
SCHEMBL2637925 0.88 KCNH2 (0.48) HDAC2HDAC3HDAC1KCNH2
SCHEMBL3133124 0.86 HDAC1 (0.43) HDAC2HDAC3HDAC1ABL1BCR
SCHEMBL2637850 0.85 HDAC1 (0.47) HDAC2HDAC3HDAC1ABL1BCR
SCHEMBL2638200 0.83 HDAC1 (0.39) HDAC2HDAC3HDAC1ABL1
SCHEMBL272439 0.82 CDK2 (0.53) HDAC2HDAC3KCNH2GSK3B
SCHEMBL2638247 0.79 HDAC1 (0.47) HDAC2HDAC3HDAC1ABL1BCR
SCHEMBL2638357 0.77 KCNH2 (0.44) HDAC2HDAC3HDAC1KCNH2
SCHEMBL2638417 0.77 TP53 (0.44) HDAC2HDAC3HDAC1ABL1BCR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2011528039-A 2011-11-10 JP claimed
WO-2010009139-A2 IMIDAZOLYL PYRIMIDINE INHIBITOR COMPOUNDS GILEAD COLORADO, INC. (US) 2010-01-21 WO claimed
WO-2010009139-A2 IMIDAZOLYL PYRIMIDINE INHIBITOR COMPOUNDS GILEAD COLORADO, INC. (US) 2010-01-21 WO disclosed