SCHEMBL2638536

SCHEMBL2638536

COc1ccc(CC(=O)Nc2ccc(S(N)(=O)=O)cc2Cl)cc1Oc1cc(Cl)cc(C#N)c1

nearest known ligand 0.60

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CA1 P00915 15/20 0.60
CA2 P00918 15/20 0.60
CA9 Q16790 10/20 0.60
CA12 O43570 8/20 0.60
CA5A P35218 2/20 0.50
CA7 P43166 2/20 0.50
CA5B Q9Y2D0 2/20 0.50
CTSD P07339 2/20 0.46
SMN1; SMN2 Q16637 1/20 0.44
RORC P51449 1/20 0.43
TP53 P04637 1/20 0.42
MAPT P10636 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4604900 0.97 CA1 (0.60) CA1CA2CA9CA12CA5A
SCHEMBL2639899 0.93 CA12 (0.50) CA1CA2CA9CA12CTSD
SCHEMBL4603625 0.92 CA1 (0.58) CA1CA2CA9CA12CA5A
SCHEMBL2639677 0.91 CA1 (0.56) CA1CA2CA9CA12CA5A
SCHEMBL2638451 0.90 CA1 (0.55) CA1CA2CA9CA12CA5A
SCHEMBL4604203 0.90 CA1 (0.56) CA1CA2CA9CA12CA5A
SCHEMBL2639756 0.90 CA1 (0.56) CA1CA2CA9CA12CA5A
SCHEMBL4604927 0.89 CA12 (0.50) CA1CA2CA9CA12CTSD
SCHEMBL4604199 0.89 CA2 (0.58) CA1CA2CA9CA12CA5A
SCHEMBL2639938 0.89 CA1 (0.53) CA1CA2CA9CA12CA5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-4810529-B2 2011-11-09 JP claimed
EP-1742908-B1 NON-NUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITORS HOFFMANN LA ROCHE (CH) 2009-11-11 EP claimed
EP-1742908-A1 NON-NUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITORS F.HOFFMANN-LA ROCHE AG (CH) 2007-01-17 EP claimed
WO-2005102989-A1 NON-NUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2005-11-03 WO claimed
EP-1742908-B1 NON-NUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITORS HOFFMANN LA ROCHE (CH) 2009-11-11 EP disclosed