SCHEMBL2638801

SCHEMBL2638801

O=C(O)CCNCc1ccc(CC=NOCc2ccc(-c3ccncc3)cc2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 16/20 0.53
ALDH1A1 P00352 2/20 0.45
ROCK2 O75116 2/20 0.38
ROCK1 Q13464 2/20 0.38
S1PR3 Q99500 2/20 0.38
RPS6KA5 O75582 1/20 0.37
MAP4K4 O95819 1/20 0.37
PRKCG P05129 1/20 0.37
PRKACA P17612 1/20 0.37
RPS6KB1 P23443 1/20 0.37
MAPK1 P28482 1/20 0.37
AKT1 P31749 1/20 0.37
GSK3A P49840 1/20 0.37
GSK3B P49841 1/20 0.37
PRKX P51817 1/20 0.37
PRKCD Q05655 1/20 0.37
PRKG2 Q13237 1/20 0.37
DYRK1A Q13627 1/20 0.37
PRKG1 Q13976 1/20 0.37
PKN2 Q16513 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4666420 0.90 S1PR1 (0.64) S1PR1
SCHEMBL2639169 0.89 S1PR1 (0.53) S1PR1
SCHEMBL2640104 0.88 S1PR1 (0.67) S1PR1S1PR3
SCHEMBL2638267 0.88 S1PR1 (0.66) S1PR1ALDH1A1S1PR3
SCHEMBL2639905 0.87 S1PR1 (0.67) S1PR1S1PR3
SCHEMBL4666263 0.84 S1PR1 (0.50) S1PR1S1PR3
SCHEMBL4663090 0.83 S1PR1 (0.52) S1PR1S1PR3
SCHEMBL2638114 0.82 S1PR1 (0.54) S1PR1S1PR3
SCHEMBL2638750 0.81 S1PR1 (0.56) S1PR1
SCHEMBL2638725 0.81 S1PR1 (0.52) S1PR1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-4700616-B2 2011-06-15 JP claimed
EP-1633336-A4 IMMUNOSUPPRESSANT COMPOUNDS AND COMPOSITIONS IRM LLC (BM) 2008-10-29 EP claimed
EP-1633336-A2 IMMUNOSUPPRESSANT COMPOUNDS AND COMPOSITIONS IRM LLC (BM) 2006-03-15 EP claimed
WO-2004103306-A2 IMMUNOSUPPRESSANT COMPOUNDS AND COMPOSITIONS IRM LLC (BM) 2004-12-02 WO claimed
EP-1633336-A4 IMMUNOSUPPRESSANT COMPOUNDS AND COMPOSITIONS IRM LLC (BM) 2008-10-29 EP disclosed
EP-1633336-A2 IMMUNOSUPPRESSANT COMPOUNDS AND COMPOSITIONS IRM LLC (BM) 2006-03-15 EP disclosed
WO-2004103306-A2 IMMUNOSUPPRESSANT COMPOUNDS AND COMPOSITIONS IRM LLC (BM) 2004-12-02 WO disclosed