SCHEMBL2639657

SCHEMBL2639657

COc1ccc(Cc2cc(OC)cc3c(-c4cccc(Cl)c4)c(C#N)c(=O)[nH]c23)c(OC)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.43
TDO2 P48775 1/20 0.43
MAPK1 P28482 1/20 0.42
HPGD P15428 4/20 0.41
HTT P42858 2/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
KDM4E B2RXH2 3/20 0.40
ALDH1A1 P00352 3/20 0.40
EGFR P00533 2/20 0.39
PIM1 P11309 1/20 0.38
GLA P06280 2/20 0.38
GAA P10253 2/20 0.38
LMNA P02545 1/20 0.37
CLK1 P49759 1/20 0.37
CLK2 P49760 1/20 0.37
DYRK1A Q13627 1/20 0.37
CLK4 Q9HAZ1 1/20 0.37
DYRK1B Q9Y463 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2639285 0.90 KCNA5 (0.46) IDO1MAPK1HPGDHTTMEN1
SCHEMBL2639613 0.79 IDO1 (0.52) IDO1TDO2MAPK1HPGDHTT
SCHEMBL3622871 0.76 EDNRB (0.45) MAPK1MEN1KMT2AKDM4EALDH1A1
SCHEMBL2639760 0.72 IDO1 (0.43) IDO1MAPK1HPGDHTTMEN1
SCHEMBL2639092 0.72 IDO1 (0.45) IDO1MAPK1HPGDHTTMEN1
SCHEMBL3621355 0.72 KCNA5 (0.46) IDO1TDO2MAPK1KDM4EALDH1A1
SCHEMBL2640067 0.72 CLK1 (0.44) IDO1MAPK1HPGDHTTMEN1
Hydrochloric Acid SCHEMBL6065024 0.72 ALDH1A1 (0.39) MAPK1HPGDMEN1KMT2ANPSR1
SCHEMBL5618029 0.71 MAPK1 (0.53) MAPK1HPGDHTTMEN1KMT2A
SCHEMBL6064429 0.70 KCNA5 (0.53) IDO1MAPK1HPGDHTTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-4794445-B2 2011-10-19 JP claimed
EP-1667973-A2 QUINOLINE POTASSIUM CHANNEL INHIBITORS Merck & Co., Inc. (US) 2006-06-14 EP claimed
WO-2005030792-A2 QUINOLINE POTASSIUM CHANNEL INHIBITORS MERCK & CO., INC. (US) 2005-04-07 WO claimed
EP-1667973-A2 QUINOLINE POTASSIUM CHANNEL INHIBITORS Merck & Co., Inc. (US) 2006-06-14 EP disclosed
WO-2005030792-A2 QUINOLINE POTASSIUM CHANNEL INHIBITORS MERCK & CO., INC. (US) 2005-04-07 WO disclosed