SCHEMBL2639671

SCHEMBL2639671

N#Cc1cc(Oc2cc(CC(=O)Nc3ccc(S(N)(=O)=O)cc3Cl)ccc2Cl)cc(C(F)(F)F)c1

nearest known ligand 0.52

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CA1 P00915 19/20 0.52
CA2 P00918 19/20 0.52
CA9 Q16790 13/20 0.52
CA12 O43570 11/20 0.52
CA5A P35218 2/20 0.49
CA7 P43166 2/20 0.49
CA5B Q9Y2D0 2/20 0.49
P2RX4 Q99571 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2638684 0.93 CA1 (0.46) CA1CA2CA9CA12CA5A
SCHEMBL2639477 0.90 P2RX4 (0.47) CA1CA2CA9CA12CA5A
SCHEMBL2638748 0.84 CA1 (0.59) CA1CA2CA9CA12CA5A
SCHEMBL2638991 0.83 CA1 (0.49) CA1CA2CA9CA12CA5A
SCHEMBL4603625 0.82 CA1 (0.58) CA1CA2CA9CA12CA5A
SCHEMBL2639829 0.82 CA1 (0.56) CA1CA2CA9CA12CA5A
SCHEMBL2639677 0.82 CA1 (0.56) CA1CA2CA9CA12CA5A
SCHEMBL2638536 0.81 CA1 (0.60) CA1CA2CA9CA12CA5A
SCHEMBL2638451 0.81 CA1 (0.55) CA1CA2CA9CA12CA5A
SCHEMBL4604900 0.81 CA1 (0.60) CA1CA2CA9CA12CA5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-4810529-B2 2011-11-09 JP claimed
EP-1742908-B1 NON-NUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITORS HOFFMANN LA ROCHE (CH) 2009-11-11 EP claimed
EP-1742908-A1 NON-NUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITORS F.HOFFMANN-LA ROCHE AG (CH) 2007-01-17 EP claimed
WO-2005102989-A1 NON-NUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2005-11-03 WO claimed
EP-1742908-B1 NON-NUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITORS HOFFMANN LA ROCHE (CH) 2009-11-11 EP disclosed