SCHEMBL2641393

SCHEMBL2641393

COC(=O)c1c(OC(C)C(N)=O)ccc2ccccc12

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NCEH1 Q6PIU2 6/20 0.58
KMT2A Q03164 2/20 0.41
MEN1 O00255 1/20 0.41
RCE1 Q9Y256 1/20 0.41
KDM4E B2RXH2 1/20 0.41
GAA P10253 1/20 0.41
HTT P42858 1/20 0.41
ALDH1A1 P00352 1/20 0.40
HPGD P15428 1/20 0.40
CYP1A2 P05177 1/20 0.40
MAPT P10636 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
GLA P06280 1/20 0.39
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA7 P43166 1/20 0.39
CA9 Q16790 1/20 0.39
CA14 Q9ULX7 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3915104 0.79 NCEH1 (0.70) NCEH1KMT2AMEN1KDM4EHTT
SCHEMBL11807725 0.79 NCEH1 (0.54) NCEH1KMT2AHPGDCYP1A2MAPT
SCHEMBL5941038 0.78 ALDH1A1 (0.49) KMT2AMEN1KDM4EGAAALDH1A1
SCHEMBL31376353 0.78 ALDH1A1 (0.49) KMT2AMEN1KDM4EGAAALDH1A1
SCHEMBL24650176 0.78 NCEH1 (0.54) NCEH1KMT2AMEN1RCE1HPGD
SCHEMBL17502745 0.78 KDM4E (0.53) NCEH1KMT2AKDM4EALDH1A1MAPT
Hydrochloric Acid SCHEMBL28705663 0.77 NCEH1 (0.53) NCEH1KMT2AMEN1RCE1HPGD
Hydrochloric Acid SCHEMBL28705662 0.77 NCEH1 (0.53) NCEH1KMT2AMEN1RCE1HPGD
Benzene SCHEMBL27947280 0.77 PPARG (0.50) KMT2AKDM4EGAAALDH1A1HPGD
SCHEMBL2556427 0.77 MAPT (0.69) NCEH1KMT2AKDM4EGAAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2438037-A1 GLYCINE B ANTAGONISTS Merz Pharma GmbH & Co. KGaA (DE) 2012-04-11 EP disclosed
WO-2010139481-A1 GLYCINE B ANTAGONISTS MERZ PHARMA GMBH & CO. KGAA (DE) 2010-12-09 WO disclosed