SCHEMBL2641795

SCHEMBL2641795

O=C(O)NCc1ccc(C=Cc2cccc(Br)n2)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.52
HPGD P15428 2/20 0.52
USP9X Q93008 1/20 0.46
CYP2D6 P10635 2/20 0.43
CYP2C9 P11712 2/20 0.43
TSHR P16473 2/20 0.43
CYP2C19 P33261 2/20 0.43
CYP1A2 P05177 1/20 0.43
HDAC6 Q9UBN7 6/20 0.42
HDAC1 Q13547 4/20 0.42
HDAC3 O15379 4/20 0.42
HDAC8 Q9BY41 4/20 0.42
HDAC2 Q92769 3/20 0.42
HDAC4 P56524 2/20 0.42
HDAC7 Q8WUI4 2/20 0.42
HDAC10 Q969S8 2/20 0.42
HDAC11 Q96DB2 2/20 0.42
HDAC9 Q9UKV0 2/20 0.42
HDAC5 Q9UQL6 2/20 0.42
MMP1 P03956 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2641788 1.00 ALDH1A1 (0.52) ALDH1A1HPGDUSP9XCYP2D6CYP2C9
SCHEMBL2641859 0.84 CYP2D6 (0.43) ALDH1A1HPGDCYP2D6CYP2C9TSHR
SCHEMBL2641932 0.84 ALDH1A1 (0.44) ALDH1A1HPGDCYP2D6CYP2C9TSHR
SCHEMBL2641898 0.84 CYP2D6 (0.43) ALDH1A1HPGDCYP2D6CYP2C9TSHR
SCHEMBL2641927 0.84 ALDH1A1 (0.44) ALDH1A1HPGDCYP2D6CYP2C9TSHR
SCHEMBL2641891 0.84 CYP2D6 (0.43) ALDH1A1HPGDCYP2D6CYP2C9TSHR
SCHEMBL2641863 0.84 CYP2D6 (0.43) ALDH1A1HPGDCYP2D6CYP2C9TSHR
SCHEMBL2641786 0.80 MAPT (0.43) ALDH1A1HPGDCYP2D6CYP2C9TSHR
SCHEMBL2641779 0.80 MAPT (0.43) ALDH1A1HPGDCYP2D6CYP2C9TSHR
SCHEMBL2641827 0.78 HDAC1 (0.44) ALDH1A1HPGDCYP2D6CYP2C9TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011141515-A1 DIAGNOSTIC AGENTS FOR AMYLOID BETA IMAGING BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2011-11-17 WO claimed
WO-2011141515-A1 DIAGNOSTIC AGENTS FOR AMYLOID BETA IMAGING BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2011-11-17 WO disclosed