SCHEMBL26425447

SCHEMBL26425447

Cc1cccc(/C=C/c2ccc3c(c2)COB3O)c1

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 12/20 0.50
PDE4A P27815 10/20 0.50
PDE4C Q08493 10/20 0.50
PDE4D Q08499 10/20 0.50
CA1 P00915 3/20 0.48
CA2 P00918 3/20 0.48
PDE3A Q14432 2/20 0.48
ALOX5 P09917 1/20 0.44
PTGS1 P23219 1/20 0.44
PTGS2 P35354 1/20 0.44
RELA Q04206 1/20 0.43
MAOB P27338 1/20 0.40
CHRM1 P11229 1/20 0.39
ADRA1A P35348 1/20 0.39
PDE1A P54750 1/20 0.39
PDE3B Q13370 1/20 0.39
PDE7A Q13946 1/20 0.39
CA12 O43570 1/20 0.38
CA9 Q16790 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26425459 0.87 PDE4B (0.61) PDE4BPDE4APDE4CPDE4DCA1
SCHEMBL26425304 0.85 PDE4B (0.56) PDE4BPDE4APDE4CPDE4DCA1
SCHEMBL26425329 0.84 RELA (0.44) PDE4BPDE4APDE4CPDE4DALOX5
SCHEMBL26425440 0.83 CA1 (0.63) PDE4BPDE4APDE4CPDE4DCA1
SCHEMBL26425445 0.83 PDE4B (0.50) PDE4BPDE4APDE4CPDE4DCA1
SCHEMBL26425448 0.83 PDE4B (0.56) PDE4BPDE4APDE4CPDE4DCA1
SCHEMBL26425450 0.80 PDE4B (0.53) PDE4BPDE4APDE4CPDE4DCA1
SCHEMBL26425601 0.80 PDE4B (0.62) PDE4BPDE4APDE4CPDE4DCA1
SCHEMBL26425455 0.80 PDE4B (0.53) PDE4BPDE4APDE4CPDE4DCA1
SCHEMBL5583348 0.78 PDE4B (0.69) PDE4BPDE4APDE4CPDE4DCA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12258360-B2 Compositions and methods for treatment of anticancer-drug resistant cancers THE GEORGE WASHINGTON UNIVERSITY (US) 2025-03-25 US disclosed
US-20230129381-A1 COMPOSITIONS AND METHODS FOR TREATMENT OF ANTICANCER-DRUG RESISTANT CANCERS THE GEORGE WASHINGTON UNIVERSITY 2023-04-27 US disclosed
US-20230129381-A1 COMPOSITIONS AND METHODS FOR TREATMENT OF ANTICANCER-DRUG RESISTANT CANCERS THE GEORGE WASHINGTON UNIVERSITY 2023-04-27 US disclosed
US-20230129381-A1 COMPOSITIONS AND METHODS FOR TREATMENT OF ANTICANCER-DRUG RESISTANT CANCERS THE GEORGE WASHINGTON UNIVERSITY 2023-04-27 US disclosed
EP-4132657-A1 COMPOSITIONS AND METHODS FOR TREATMENT OF ANTICANCER-DRUG RESISTANT CANCERS The George Washington University (US) 2023-02-15 EP disclosed
CN-111333672-B Sterol regulatory element binding protein and acidic nucleoplasm DNA binding protein-1 inhibitor, and preparation method and application thereof 中国医学科学院放射医学研究所 2022-11-08 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12258360-B2 Compositions and methods for treatment of anticancer-drug resistant cancers TP53, ANXA5, MCL1 PDE4B 2973/4885PDE4A 3402/4885PDE4C 2702/4885
US-20230129381-A1 COMPOSITIONS AND METHODS FOR TREATMENT OF ANTICANCER-DRUG RESISTANT CANCERS TP53, ANXA5, MCL1 PDE4B 2973/4885PDE4A 3402/4885PDE4C 2702/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.