SCHEMBL2643846

SCHEMBL2643846

O=C(O)CC1c2ccccc2C(=O)N1Cc1ccc(F)cc1

nearest known ligand 0.56

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.56
MDM2 Q00987 3/20 0.48
MEN1 O00255 1/20 0.45
TSHR P16473 1/20 0.45
MAPK1 P28482 1/20 0.45
KMT2A Q03164 1/20 0.45
CASP3 P42574 1/20 0.44
WDR5 P61964 1/20 0.43
KCNA5 P22460 1/20 0.43
KCNH2 Q12809 1/20 0.43
ATM Q13315 1/20 0.42
PRMT5 O14744 2/20 0.42
WDR77 Q9BQA1 2/20 0.42
TOP1 P11387 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4476753 0.91 MAPT (0.53) MAPTMDM2MEN1TSHRMAPK1
SCHEMBL2644438 0.88 MAPT (0.54) MAPTMDM2MEN1TSHRMAPK1
SCHEMBL2643388 0.85 MAPT (0.55) MAPTMDM2MEN1KMT2AKCNA5
SCHEMBL30296312 0.84 MEN1 (0.51) MAPTMDM2MEN1TSHRMAPK1
SCHEMBL2643804 0.84 MEN1 (0.51) MAPTMDM2MEN1TSHRMAPK1
SCHEMBL2643902 0.81 MAPT (0.50) MAPTMDM2MEN1TSHRMAPK1
SCHEMBL27725675 0.81 MAPT (0.50) MAPTMDM2MEN1TSHRMAPK1
SCHEMBL4486492 0.78 FFAR1 (0.49) MAPTMEN1TSHRMAPK1KMT2A
SCHEMBL2643221 0.78 MAPT (0.50) MAPTMDM2
SCHEMBL2645468 0.77 MEN1 (0.51) MAPTMDM2MEN1TSHRMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8796313-B2 Substituted dihydroisoindolones as allosteric modulators of glucokinase JANSSEN PHARMACEUTICA N.V. (BE) 2014-08-05 US disclosed
CN-101316836-A Substituted dihydroisoindolones as allosteric modulators of glucokinase JANSSEN PHARMACEUTICA NV (BE) 2008-12-03 CN disclosed
US-20070099930-A1 Substituted Dihydroisoindolones As Allosteric Modulators of Glucokinase JANSSEN PHARMACEUTICA N.V. (BE) 2007-05-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070099930-A1 Substituted Dihydroisoindolones As Allosteric Modulators of Glucokinase GCK, GCKR, GPR119 MAPT 3322/4885MDM2 2023/4885MEN1 4234/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.