SCHEMBL2644976

SCHEMBL2644976

CCS(=O)(=O)c1ccc(Oc2cc(Oc3c(F)cccc3C(N)=O)c3nc(-c4ccccn4)[nH]c3c2)cn1

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GCK P35557 13/20 0.42
CBFB Q13951 6/20 0.39
PARP1 P09874 1/20 0.39
DHODH Q02127 1/20 0.39
PARP2 Q9UGN5 1/20 0.39
ALDH1A1 P00352 1/20 0.36
TP53 P04637 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
HPGD P15428 1/20 0.36
ALOX15 P16050 1/20 0.36
CYP2C19 P33261 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
HSD17B10 Q99714 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2645184 0.93 DHODH (0.40) GCKCBFBPARP1DHODHPARP2
SCHEMBL2645652 0.92 DHODH (0.37) GCKPARP1DHODHPARP2CYP3A4
SCHEMBL2644582 0.92 CBFB (0.44) GCKCBFBALDH1A1TP53CYP3A4
SCHEMBL2644898 0.88 GCK (0.53) GCK
SCHEMBL2645885 0.86 GCK (0.40) GCKCBFBALDH1A1TP53CYP3A4
SCHEMBL2645338 0.86 CBFB (0.45) GCKCBFBALDH1A1TP53CYP3A4
SCHEMBL2645888 0.84 CBFB (0.43) GCKCBFBALDH1A1TP53CYP3A4
SCHEMBL2643868 0.83 GCK (0.37) GCKCBFBDHODHCYP3A4CYP2C19
SCHEMBL1657673 0.83 GCK (0.45) GCKCBFBPARP1DHODHPARP2
SCHEMBL2646321 0.83 CBFB (0.43) GCKCBFBALDH1A1TP53CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1702919-B1 NOVEL 2-HETEROARYL-SUBSTITUTED BENZIMIDAZOLE DERIVATIVE MSD KK (JP) 2012-05-30 EP disclosed
EP-1702919-A1 NOVEL 2-HETEROARYL-SUBSTITUTED BENZIMIDAZOLE DERIVATIVE BANYU PHARMACEUTICAL CO., LTD. (JP) 2006-09-20 EP disclosed