SCHEMBL2646405

SCHEMBL2646405

COC(OC)c1ccncc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.46
CYP2C19 P33261 2/20 0.46
SLC6A2 P23975 2/20 0.42
SLC6A4 P31645 2/20 0.42
SLC6A3 Q01959 2/20 0.42
CYP17A1 P05093 2/20 0.40
CYP19A1 P11511 2/20 0.39
GAA P10253 1/20 0.38
KMT2A Q03164 2/20 0.37
MEN1 O00255 1/20 0.37
MAPT P10636 2/20 0.36
LMNA P02545 1/20 0.36
ALDH1A1 P00352 2/20 0.36
HPGD P15428 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
KDM4E B2RXH2 1/20 0.35
NPC1 O15118 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8955219 0.80 CA12 (0.35) CYP3A4CYP2C19SLC6A4ALDH1A1KDM4E
SCHEMBL9129250 0.77 SLC6A2 (0.46) CYP3A4CYP2C19SLC6A2SLC6A4SLC6A3
SCHEMBL17011305 0.77 SLC6A2 (0.46) CYP3A4CYP2C19SLC6A2SLC6A4SLC6A3
SCHEMBL12784512 0.77 SLC6A2 (0.46) CYP3A4CYP2C19SLC6A2SLC6A4SLC6A3
SCHEMBL8349612 0.75 CYP3A4 (0.43) CYP3A4CYP2C19SLC6A2SLC6A4SLC6A3
SCHEMBL6632699 0.75 CYP3A4 (0.43) CYP3A4CYP2C19SLC6A2SLC6A4SLC6A3
SCHEMBL623356 0.73 PTGS2 (0.44) CYP3A4CYP2C19SLC6A2SLC6A4SLC6A3
SCHEMBL26689 0.72 KMT2A (0.44) KMT2AMEN1MAPTLMNASMN1; SMN2
SCHEMBL21162070 0.72 TSHR (0.34) CYP3A4CYP17A1ALDH1A1
SCHEMBL15350067 0.72 TSHR (0.34) CYP3A4CYP17A1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 64 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112661694-B Preparation method of 4- (dimethoxymethyl) -piperidine 西安凯立新材料股份有限公司 2023-04-11 CN claimed
CN-112661694-A Preparation method of 4- (dimethoxymethyl) -piperidine 西安凯立新材料股份有限公司 2021-04-16 CN claimed
CN-102344440-B Anticoccidial compound for livestock and poultry and preparation method thereof CHINA ANIMAL HUSBANDRY INDUSTRY CO LTD 2013-10-30 CN claimed
CN-102408413-B Anticoccidial compound, and preparation method and use thereof CHINA ANIMAL HUSBANDRY INDUSTRY CO LTD 2013-08-14 CN claimed
CN-102311425-B Anticoccidiosis compound and preparation method as well as application thereof CHINA ANIMAL HUSBANDRY INDUSTRY CO LTD 2013-06-05 CN claimed
CN-102408413-A Anticoccidial compound and preparation method and application thereof CHINA ANIMAL HUSBANDRY INDUSTRY CO LTD 2012-04-11 CN claimed
CN-102344440-A Anticoccidial compound for livestock and poultry and preparation method thereof CHINA ANIMAL HUSBANDRY INDUSTRY CO LTD 2012-02-08 CN claimed
CN-102311425-A Anticoccidiosis compound and preparation method as well as application thereof CHINA ANIMAL HUSBANDRY INDUSTRY CO LTD 2012-01-11 CN claimed
WO-2024063576-A1 NOVEL QUINAZOLINE COMPOUND AS KRAS INHIBITOR 일동제약(주) 2024-03-28 WO disclosed
CN-112661694-B Preparation method of 4- (dimethoxymethyl) -piperidine 西安凯立新材料股份有限公司 2023-04-11 CN disclosed
CN-112661694-B Preparation method of 4- (dimethoxymethyl) -piperidine 西安凯立新材料股份有限公司 2023-04-11 CN disclosed
CN-112661694-A Preparation method of 4- (dimethoxymethyl) -piperidine 西安凯立新材料股份有限公司 2021-04-16 CN disclosed
CN-112661694-A Preparation method of 4- (dimethoxymethyl) -piperidine 西安凯立新材料股份有限公司 2021-04-16 CN disclosed
CN-107667092-A Formylated N Hete rocyclic derivatives as FGFR4 inhibitor 诺华股份有限公司 2018-02-06 CN disclosed
EP-0854870-A1 SUBSTITUTED IMIDAZOLES HAVING ANTI-CANCER AND CYTOKINE INHIBITORY ACTIVITY Merck & Co., Inc. (US) 1998-07-29 EP disclosed
US-5776954-A GLUCAGON ANTAGONISTS MERCK & CO., INC. (US) 1998-07-07 US disclosed
US-5717100-A Substituted imidazoles having anti-cancer and cytokine inhibitory activity MERCK & CO., INC. (US) 1998-02-10 US disclosed
WO-1997012876-A9 SUBSTITUTED IMIDAZOLES HAVING ANTI-CANCER AND CYTOKINE INHIBITORY ACTIVITY 1997-09-18 WO disclosed
WO-1997016442-A1 SUBSTITUTED PYRIDYL PYRROLES, COMPOSITIONS CONTAINING SUCH COMPOUNDS AND METHODS OF USE MERCK & CO., INC. (US) 1997-05-09 WO disclosed
WO-1997012876-A1 SUBSTITUTED IMIDAZOLES HAVING ANTI-CANCER AND CYTOKINE INHIBITORY ACTIVITY MERCK & CO., INC. (US) 1997-04-10 WO disclosed