SCHEMBL2646501

SCHEMBL2646501

Fc1ccc(Oc2cc(Oc3cccnc3)cc3[nH]c(-c4cnccn4)nc23)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CBFB Q13951 3/20 0.41
CYP19A1 P11511 1/20 0.41
METAP2 P50579 1/20 0.40
CHEK2 O96017 1/20 0.39
CYP11B1 P15538 2/20 0.38
FFAR4 Q5NUL3 2/20 0.38
CYP11B2 P19099 1/20 0.38
GRM5 P41594 1/20 0.37
DHODH Q02127 2/20 0.36
LMNA P02545 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
LTA4H P09960 1/20 0.35
WNT1 P04628 1/20 0.35
TGFBR1 P36897 1/20 0.35
GCK P35557 1/20 0.35
ALDH1A1 P00352 1/20 0.35
TP53 P04637 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
HPGD P15428 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2645922 0.91 CBFB (0.52) CBFBMETAP2GRM5GCKALDH1A1
SCHEMBL2646787 0.88 CBFB (0.40) CBFBCYP19A1CHEK2CYP11B1FFAR4
SCHEMBL2645836 0.88 CHEK2 (0.42) CBFBCYP19A1CHEK2CYP11B1FFAR4
SCHEMBL2644929 0.86 CHEK2 (0.41) CBFBCYP19A1CHEK2CYP11B1FFAR4
SCHEMBL2646329 0.86 CYP2E1 (0.38) CBFBCYP19A1CHEK2CYP11B1FFAR4
SCHEMBL2645371 0.85 CBFB (0.38) CBFBCYP19A1CHEK2CYP11B1FFAR4
SCHEMBL2646095 0.84 CHEK2 (0.36) CBFBCYP19A1CHEK2CYP11B1FFAR4
SCHEMBL2645553 0.83 CBFB (0.55) CBFBMETAP2GRM5LMNAALDH1A1
SCHEMBL2646752 0.83 CHEK2 (0.36) CBFBCYP19A1CHEK2CYP11B1FFAR4
SCHEMBL2644100 0.82 CBFB (0.51) CBFBMETAP2GRM5LMNATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1702919-B1 NOVEL 2-HETEROARYL-SUBSTITUTED BENZIMIDAZOLE DERIVATIVE MSD KK (JP) 2012-05-30 EP disclosed
EP-1702919-A1 NOVEL 2-HETEROARYL-SUBSTITUTED BENZIMIDAZOLE DERIVATIVE BANYU PHARMACEUTICAL CO., LTD. (JP) 2006-09-20 EP disclosed