SCHEMBL264729

SCHEMBL264729

FC(F)(F)c1cc(Br)ccc1Cl

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.47
HTR3E A5X5Y0 1/20 0.47
HTR3B O95264 1/20 0.47
HTR3A P46098 1/20 0.47
HTR3D Q70Z44 1/20 0.47
HTR3C Q8WXA8 1/20 0.47
KDR P35968 1/20 0.47
KDM1A O60341 2/20 0.46
NT5E P21589 1/20 0.46
NOTUM Q6P988 7/20 0.44
LMNA P02545 1/20 0.43
TP53 P04637 1/20 0.43
MAPT P10636 1/20 0.43
THRB P10828 1/20 0.43
RAPGEF4 Q8WZA2 1/20 0.42
PDK1 Q15118 1/20 0.42
NPFFR2 Q9Y5X5 3/20 0.41
NPFFR1 Q9GZQ6 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29707579 1.00 IDO1 (0.47) IDO1HTR3EHTR3BHTR3AHTR3D
SCHEMBL5779231 0.83 NT5E (0.40) IDO1HTR3EHTR3BHTR3AHTR3D
SCHEMBL31342658 0.83 NT5E (0.40) IDO1HTR3EHTR3BHTR3AHTR3D
SCHEMBL585377 0.82 NT5E (0.46) IDO1HTR3EHTR3BHTR3AHTR3D
SCHEMBL29589267 0.82 NT5E (0.46) IDO1HTR3EHTR3BHTR3AHTR3D
SCHEMBL2043993 0.79 NT5E (0.38) IDO1HTR3EHTR3BHTR3AHTR3D
SCHEMBL6267032 0.78 KDM1A (0.50) KDM1ANT5ENOTUMNPFFR2NPFFR1
SCHEMBL30864218 0.78 KDM1A (0.50) KDM1ANT5ENOTUMNPFFR2NPFFR1
SCHEMBL12791524 0.77 PTGDR2 (0.42) NT5ETP53MAPT
SCHEMBL4209652 0.77 KDM1A (0.46) KDM1ANT5ENPFFR2NPFFR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 367 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118652170-A New synthesis method of 5-bromo-2-chlorobenzoic acid 宁夏法安德药业有限公司 2024-09-17 CN claimed
CN-115819353-B Method for preparing 2-arylamino benzimidazole and N1-aryl-2-amino benzimidazole 长沙晶易医药科技股份有限公司 2023-06-30 CN claimed
US-20260124309-A1 STAT6 DEGRADERS AND USES THEREOF KYMERA THERAPEUTICS INC (US) 2026-05-07 US disclosed
US-12577257-B2 Heterocyclic compounds HOFFMANN-LA ROCHE INC. (US) 2026-03-17 US disclosed
US-12410212-B2 Cyclic compound having selective KRAS inhibitory effect on HRAS and NRAS CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2025-09-09 US disclosed
EP-4603105-A1 PHARMACEUTICAL COMPOSITION CONTAINING CYCLIC COMPOUND HAVING SELECTIVE KRAS INHIBITORY EFFECT AGAINST HRAS AND NRAS CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2025-08-20 EP disclosed
EP-4592308-A1 CYCLIC COMPOUND HAVING SELECTIVE KRAS INHIBITORY EFFECT ON HRAS AND NRAS CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2025-07-30 EP disclosed
US-20250230193-A1 CYCLIC COMPOUND HAVING SELECTIVE KRAS INHIBITORY EFFECT ON HRAS AND NRAS CHUGAI PHARMACEUTICAL CO LTD (JP) 2025-07-17 US disclosed
CN-120202211-A Cyclic compounds having selective KRAS inhibition over HRAS and NRAS 中外制药株式会社 2025-06-24 CN disclosed
US-12286432-B2 Fluorinated tetrahydronaphthyridinyl nonanoic acid derivatives and uses thereof OCUTERRA THERAPEUTICS, INC. (US) 2025-04-29 US disclosed
CN-119731195-A Cyclic compounds having selective inhibition of KRAS over HRAS and NRAS 中外制药株式会社 2025-03-28 CN disclosed
US-4396770-A ANALGESICS, PSYCHOSIS HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1983-08-02 US disclosed
EP-0020018-B1 CHROMAN DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM BEECHAM GROUP PLC (GB) 1983-06-01 EP disclosed
EP-0063799-A2 1-(3-(6-fluoro-1,2-benzisoxasol-3-yl)propyl)-4-hydroxy-4-phenylpiperidines, a process for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1982-11-03 EP disclosed
US-4303656-A ANOREXIC AGENTS BEECHAM GROUP LIMITED (GB) 1981-12-01 US disclosed
EP-0020018-A1 Chroman derivatives, processes for their preparation and pharmaceutical compositions containing them BEECHAM GROUP PLC (GB) 1980-12-10 EP disclosed
US-4213989-A 3-TRIFLUOROMETHYL GROUP ON PHENYL ROUSSEL UCLAF (FR) 1980-07-22 US disclosed
US-4155940-A M-Bromo-benzotrifluorides BAYER AKTIENGESELLSCHAFT (DE) 1979-05-22 US disclosed
US-4076821-A 4,4-Diphenylcycloalkylpiperidines and psychotropic compositions thereof YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JA) 1978-02-28 US disclosed
US-3947460-A SEDATIVES-HYPNOTIC, TRANQUILIZER SANDOZ, INC. (US) 1976-03-30 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260124309-A1 STAT6 DEGRADERS AND USES THEREOF STAT6, NCOR2, NCOR1 IDO1 173/4885HTR3E 1849/4885HTR3B 1404/4885
US-12410212-B2 Cyclic compound having selective KRAS inhibitory effect on HRAS and NRAS KRAS, HRAS, NRAS IDO1 4447/4885HTR3E 4666/4885HTR3B 4507/4885
US-12286432-B2 Fluorinated tetrahydronaphthyridinyl nonanoic acid derivatives and uses thereof FFAR3, FFAR2, FFAR1 IDO1 2603/4885HTR3E 1128/4885HTR3B 999/4885
US-20250230193-A1 CYCLIC COMPOUND HAVING SELECTIVE KRAS INHIBITORY EFFECT ON HRAS AND NRAS KRAS, HRAS, NRAS IDO1 4447/4885HTR3E 4666/4885HTR3B 4507/4885
US-12577257-B2 Heterocyclic compounds H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16, CBR1, CBR3 IDO1 3471/4885HTR3E 1678/4885HTR3B 1565/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.