SCHEMBL2647293

SCHEMBL2647293

C1=CC2NCCCC2CCC1

nearest known ligand 0.32

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
EPAS1 Q99814 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10757117 0.91 EPAS1 (0.32) EPAS1
SCHEMBL8603606 0.85 EPAS1 (0.34) EPAS1
SCHEMBL22460801 0.84 EPAS1 (0.32) EPAS1
SCHEMBL17881911 0.83 EPAS1 (0.32) EPAS1
SCHEMBL2292798 0.82
SCHEMBL21722414 0.77
SCHEMBL10914129 0.77
SCHEMBL8901938 0.76 CHRNB2 (0.30)
SCHEMBL9726321 0.72 EPAS1 (0.31) EPAS1
SCHEMBL1434651 0.72 EPAS1 (0.31) EPAS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 17 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1463715-A1 NOVEL GLUCAGON ANTAGONISTS NOVO NORDISK A/S (DK) 2004-10-06 EP disclosed
WO-2003048109-A1 NOVEL GLUCAGON ANTAGONISTS NOVO NORDISK A/S (DK) 2003-06-12 WO disclosed
EP-1124830-A1 PYRIMIDIN-4-ENAMINE AS FUNGICIDE Syngenta Participations AG (CH) 2001-08-22 EP disclosed
EP-1087939-A1 PROCESS FOR PREPARATION OF PYRIMIDINONE DERIVATIVES Syngenta Participations AG (CH) 2001-04-04 EP disclosed
EP-1015434-A2 NOVEL PYRIMIDIN-4-ONE AND PYRIMIDIN-4-THIONE AS FUNGICIDE Novartis AG (CH) 2000-07-05 EP disclosed
EP-1015435-A1 PYRIMIDIN-2-OXY-4-ONE AND PYRIMIDIN-2-OXY-4-THIONE DERIVATIVES Novartis AG (CH) 2000-07-05 EP disclosed
WO-2000031082-A1 PYRIMIDIN-4-ENAMINE AS FUNGICIDE SYNGENTA PARTICIPATIONS AG (CH) 2000-06-02 WO disclosed
EP-0993432-A1 PROCESS FOR THE PREPARATION OF TRIFLUOROMETHYL ACETOPHENONE Novartis AG (CH) 2000-04-19 EP disclosed
WO-1999067202-A1 PROCESS FOR PREPARATION OF PYRIMIDINONE DERIVATIVES SYNGENTA PARTICIPATIONS AG . (CH) 1999-12-29 WO disclosed
EP-0912499-A1 PESTICIDES Novartis AG (CH) 1999-05-06 EP disclosed
WO-1999014202-A2 NOVEL PYRIMIDIN-4-ONE AND PYRIMIDIN-4-THIONE AS FUNGICIDE NOVARTIS AG (CH) 1999-03-25 WO disclosed
WO-1999011631-A1 PYRIMIDIN-2-OXY-4-ONE AND PYRIMIDIN-2-OXY-4-THIONE DERIVATIVES NOVARTIS AG (CH) 1999-03-11 WO disclosed
EP-0888359-A1 PYRIMIDIN-4-ONE DERIVATIVES AS PESTICIDE Novartis AG (CH) 1999-01-07 EP disclosed
WO-1998058895-A1 PROCESS FOR THE PREPARATION OF TRIFLUOROMETHYL ACETOPHENONE NOVARTIS AG (CH) 1998-12-30 WO disclosed
WO-1997047592-A1 PESTICIDES NOVARTIS AG (CH) 1997-12-18 WO disclosed
WO-1997033890-A1 PYRIMIDIN-4-ONE DERIVATIVES AS PESTICIDE NOVARTIS AG (CH) 1997-09-18 WO disclosed
WO-1997014688-A1 A PROCESS FOR THE PREPARATION OF α-CHLOROMETHYLPHENYLACETIC ACID DERIVATIVES NOVARTIS AG (CH) 1997-04-24 WO disclosed