SCHEMBL2648829

SCHEMBL2648829

CON=Cc1ccc2c(c1)ncn2-c1cccc(Br)c1

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
FGFR1 P11362 10/20 0.44
SIK1 P57059 2/20 0.43
SIK2 Q9H0K1 2/20 0.43
SIK3 Q9Y2K2 2/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
KDR P35968 1/20 0.41
SRC P12931 3/20 0.40
ALDH1A1 P00352 1/20 0.39
HPGD P15428 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2649581 0.83 GABRA1 (0.43) FGFR1KDRSRCALDH1A1HPGD
SCHEMBL2648797 0.82 HPGD (0.47) FGFR1KDRALDH1A1HPGD
SCHEMBL2658127 0.81 FGFR1 (0.40) FGFR1KDRSRCALDH1A1
SCHEMBL1761712 0.81 GABRA1 (0.44) FGFR1KDRSRCALDH1A1HPGD
SCHEMBL2649006 0.80 FGFR1 (0.67) FGFR1SIK1SIK2SIK3MEN1
SCHEMBL1761821 0.80 FGFR1 (0.45) FGFR1KDRSRC
SCHEMBL2650162 0.80 FGFR1 (0.43) FGFR1KDRSRCALDH1A1HPGD
SCHEMBL2648539 0.80 KDR (0.41) FGFR1KDRSRCALDH1A1HPGD
SCHEMBL12415699 0.79 FGFR1 (0.54) FGFR1SIK1SIK2SIK3MEN1
SCHEMBL2648738 0.79 GABRA1 (0.41) FGFR1KDRSRCALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0821682-B1 BENZIMIDAZOLE COMPOUNDS AND THEIR USE AS MODULATORS OF THE GABA-A RECEPTOR COMPLEX NEUROSEARCH AS (DK) 2000-07-19 EP disclosed
US-5922725-A Benzimidazole compounds and their use as modulators of the GABAA receptor complex NEUROSEARCH A/S (DK) 1999-07-13 US disclosed
EP-0821682-A1 BENZIMIDAZOLE COMPOUNDS AND THEIR USE AS MODULATORS OF THE GABA A? RECEPTOR COMPLEX NEUROSEARCH A/S (DK) 1998-02-04 EP disclosed
WO-1996033191-A1 BENZIMIDAZOLE COMPOUNDS AND THEIR USE AS MODULATORS OF THE GABAA RECEPTOR COMPLEX NEUROSEARCH A/S (DK) 1996-10-24 WO disclosed