SCHEMBL2651407

SCHEMBL2651407

COc1ccc2cc(C=NN)ccc2c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 4/20 0.48
CYP2A6 P11509 1/20 0.48
CYP19A1 P11511 2/20 0.47
NQO2 P16083 2/20 0.46
CHRM5 P08912 1/20 0.46
RELA Q04206 1/20 0.44
CYP1A1 P04798 3/20 0.44
CYP1B1 Q16678 3/20 0.44
ESR1 P03372 2/20 0.44
PTGS2 P35354 2/20 0.44
ABL1 P00519 1/20 0.44
TTR P02766 1/20 0.44
ABCB1 P08183 1/20 0.44
ALOX5 P09917 1/20 0.44
BCR P11274 1/20 0.44
TUBB4A P04350 1/20 0.44
TUBB P07437 1/20 0.44
TUBA3C P0DPH7 1/20 0.44
AHR P35869 1/20 0.44
TUBA1B P68363 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20691469 0.83 CYP1A2 (0.50) CYP1A2CYP2A6CYP19A1NQO2CHRM5
SCHEMBL4672669 0.83 CYP1A2 (0.50) CYP1A2CYP2A6CYP19A1NQO2CHRM5
SCHEMBL4672666 0.83 CYP1A2 (0.50) CYP1A2CYP2A6CYP19A1NQO2CHRM5
SCHEMBL3971293 0.82 GRIN2D (0.58) CYP1A2CYP2A6RELAPTGS2MAOA
SCHEMBL3657928 0.82 GRIN2D (0.58) CYP1A2CYP2A6RELAPTGS2MAOA
SCHEMBL31499212 0.81 KDM4E (0.61) CYP1A2CYP2A6CYP19A1NQO2CHRM5
SCHEMBL31182402 0.79 CHRM5 (0.72) CYP1A2CYP19A1NQO2CHRM5RELA
SCHEMBL14950238 0.79 CHRM5 (0.72) CYP1A2CYP19A1NQO2CHRM5RELA
SCHEMBL27885399 0.79 CHRM5 (0.72) CYP1A2CYP19A1NQO2CHRM5RELA
SCHEMBL23934771 0.79 CYP1A2 (0.46) CYP1A2CYP2A6CYP19A1NQO2CHRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6613942-B1 Nonpeptide; 4-hydroxy benzoic acid hydrazides NOVO NORDISK A/S (DK) 2003-09-02 US disclosed
EP-0994848-A1 GLUCAGON ANTAGONISTS/INVERSE AGONISTS NOVO NORDISK A/S (DK) 2000-04-26 EP disclosed
WO-1999001423-A1 GLUCAGON ANTAGONISTS/INVERSE AGONISTS NOVO NORDISK A/S (DK) 1999-01-14 WO disclosed