SCHEMBL2656961

SCHEMBL2656961

O=C(NC1CC1)c1ccc2c(=O)[nH]cnc2c1

nearest known ligand 0.59

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.59
LMNA P02545 1/20 0.59
SMYD3 Q9H7B4 7/20 0.54
ALDH1A1 P00352 3/20 0.48
HPGD P15428 2/20 0.48
PARP1 P09874 2/20 0.48
CHEK1 O14757 1/20 0.48
PIM1 P11309 1/20 0.48
RPS6KA3 P51812 1/20 0.48
KMT2A Q03164 2/20 0.47
MAPT P10636 1/20 0.47
HTT P42858 1/20 0.47
SLC2A1 P11166 1/20 0.47
MAPK14 Q16539 1/20 0.47
RAB9A P51151 2/20 0.44
MEN1 O00255 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3083852 0.86 MAPK14 (0.66) MAPK14
SCHEMBL6775104 0.83 NPC1 (0.45) NPC1LMNAALDH1A1HPGDKMT2A
SCHEMBL2116618 0.82 HDAC6 (0.61) ALDH1A1PARP1CHEK1PIM1RPS6KA3
SCHEMBL263941 0.80 PARP1 (0.58) ALDH1A1PARP1CHEK1PIM1RPS6KA3
SCHEMBL3984993 0.77 NPC1 (0.64) NPC1LMNASMYD3ALDH1A1HPGD
SCHEMBL30265317 0.76 NPC1 (0.81) NPC1LMNASMYD3ALDH1A1HPGD
SCHEMBL30205640 0.76 PARP1 (0.57) ALDH1A1PARP1CHEK1PIM1RPS6KA3
SCHEMBL13908150 0.76 SLC2A1 (0.77) ALDH1A1PARP1CHEK1PIM1RPS6KA3
SCHEMBL2315757 0.76 PARP1 (0.57) ALDH1A1PARP1CHEK1PIM1RPS6KA3
SCHEMBL265032 0.75 PARP1 (0.56) ALDH1A1PARP1CHEK1PIM1RPS6KA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2001875-A2 GLUCOKINASE ACTIVATORS Takeda San Diego, Inc. (US) 2008-12-17 EP claimed
WO-2007104034-A2 GLUCOKINASE ACTIVATORS TAKEDA SAN DIEGO, INC. (US) 2007-09-13 WO claimed