SCHEMBL2658154

SCHEMBL2658154

N=C=NCCN1CCOCC1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.51
SMN1; SMN2 Q16637 3/20 0.42
ALDH1A1 P00352 2/20 0.42
KEAP1 Q14145 1/20 0.42
KDM4E B2RXH2 1/20 0.42
GLA P06280 1/20 0.38
RXFP1 Q9HBX9 1/20 0.36
HPGD P15428 1/20 0.35
DUSP3 P51452 1/20 0.35
USP2 O75604 1/20 0.34
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA9 Q16790 1/20 0.34
POLB P06746 1/20 0.34
SIGMAR1 Q99720 1/20 0.34
CYP2D6 P10635 1/20 0.33
HSD17B10 Q99714 1/20 0.33
MAPK1 P28482 1/20 0.33
HIF1A Q16665 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15253474 0.88 SMN1; SMN2 (0.48) CYP1A2SMN1; SMN2ALDH1A1KEAP1KDM4E
SCHEMBL15153786 0.87 CYP1A2 (0.42) CYP1A2SMN1; SMN2ALDH1A1KDM4EGLA
SCHEMBL11586872 0.83 CYP1A2 (0.64) CYP1A2SMN1; SMN2ALDH1A1KEAP1KDM4E
SCHEMBL2256760 0.79 CYP1A2 (0.51) CYP1A2SMN1; SMN2ALDH1A1KEAP1KDM4E
SCHEMBL838431 0.79 CYP1A2 (0.51) CYP1A2SMN1; SMN2ALDH1A1KEAP1KDM4E
SCHEMBL14376932 0.79 CYP1A2 (0.51) CYP1A2SMN1; SMN2ALDH1A1KEAP1KDM4E
SCHEMBL3281225 0.78 USP2 (0.37) CYP1A2SMN1; SMN2ALDH1A1KEAP1KDM4E
SCHEMBL9846522 0.77 ALDH1A1 (0.45) CYP1A2SMN1; SMN2ALDH1A1KDM4EGLA
SCHEMBL10352983 0.76 CYP1A2 (0.57) CYP1A2SMN1; SMN2ALDH1A1KEAP1KDM4E
SCHEMBL18434868 0.76 KDM4E (0.46) CYP1A2SMN1; SMN2ALDH1A1KEAP1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 100 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025044684-A1 PREPARATION METHOD FOR HUMAN BIOLOGICAL CORNEAL STROMA, AND USE OF HUMAN BIOLOGICAL CORNEAL STROMA 山东第一医科大学附属眼科研究所(山东省眼科研究所、山东第一医科大学附属青岛眼科医院) 2025-03-06 WO claimed
CN-117065098-B Preparation method and application of human biological cornea stroma 山东第一医科大学附属眼科研究所(山东省眼科研究所、山东第一医科大学附属青岛眼科医院) 2024-11-22 CN claimed
WO-2024059495-A1 METHODS OF PREPARING ERGOLINE ANALOGS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2024-03-21 WO claimed
CN-117065098-A Preparation method and application of human biological cornea stroma 山东第一医科大学附属眼科研究所(山东省眼科研究所、山东第一医科大学附属青岛眼科医院) 2023-11-17 CN claimed
US-20220298226-A1 METHACRYLATED COLLAGEN JELLAGEN LTD (GB) 2022-09-22 US claimed
EP-3500646-A1 CHEMISTRY FOR FINES FIXING AND WATER CONTROL Commonwealth Scientific and Industrial Research Organisation (AU) 2019-06-26 EP claimed
WO-2018032051-A1 CHEMISTRY FOR FINES FIXING AND WATER CONTROL COMMONWEALTH SCIENTIFIC AND INDUSTRIAL RESEARCH ORGANISATION (AU) 2018-02-22 WO claimed
CN-104755472-A Isotopologues of 3-(5-amino-2-methyl-4-oxoquinazolin-3(4H)-yl)piperidine-2,6-dione and methods of preparation thereof CELGENE CORP 2015-07-01 CN claimed
US-4738843-A Anti-tumor substance of immunoglobulin and melphalan and process for producing the same KUREHA KAGAKU KOGYO KABUSHIKI KAISHA (JP) 1988-04-19 US claimed
EP-0004570-B1 THIOL ESTERS, PROCESS FOR THEIR PREPARATION, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND A PROCESS FOR PREPARING CEPHALOSPORIN COMPOUNDS USING THE SAME Asahi Kasei Kogyo Kabushiki Kaisha (JP) 1982-04-14 EP claimed
WO-2025044684-A1 PREPARATION METHOD FOR HUMAN BIOLOGICAL CORNEAL STROMA, AND USE OF HUMAN BIOLOGICAL CORNEAL STROMA 山东第一医科大学附属眼科研究所(山东省眼科研究所、山东第一医科大学附属青岛眼科医院) 2025-03-06 WO disclosed
WO-2024259257-A2 CARRIER-BASE COMPLEXES AND METHODS OF USE THEREOF THE METHODIST HOSPITAL (US) 2024-12-19 WO disclosed
EP-4472969-A1 PROCESS FOR THE SYNTHESIS OF PYRAZOLYL DERIVATIVES USEFUL AS ANTI-CANCER AGENTS Novartis AG (CH) 2024-12-11 EP disclosed
CN-117065098-B Preparation method and application of human biological cornea stroma 山东第一医科大学附属眼科研究所(山东省眼科研究所、山东第一医科大学附属青岛眼科医院) 2024-11-22 CN disclosed
CN-118871436-A Synthesis of pyrazolyl derivatives useful as anticancer agents 诺华股份有限公司 2024-10-29 CN disclosed
EP-0071891-A2 New cephem compounds and processes for preparation thereof FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1983-02-16 EP disclosed
EP-0010313-B1 3,7-DISUBSTITUTED-2- OR -3-CEPHEM-4-CARBOXYLIC ACID COMPOUNDS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND PROCESSES FOR THE PREPARATION THEREOF FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1983-01-26 EP disclosed
EP-0062328-A2 Novel penicillin and cephalosporin compounds, a process for preparing the same and antibacterial composition containing the novel compounds Eisai Co., Ltd. (JP) 1982-10-13 EP disclosed
EP-0001125-B1 CEPHALOSPORIN DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1981-11-11 EP disclosed
EP-0018360-B1 N-(5-METHOXYBENZOFURAN-2-YLCARBONYL)-N'-BENZYLPIPERAZINE AND PROCESS FOR ITS PREPARATION HOECHST AKTIENGESELLSCHAFT (DE) 1981-09-30 EP disclosed