SCHEMBL2658932

SCHEMBL2658932

CCOC(=O)c1c[nH]c2c(F)c(C(F)(F)F)ccc2c1=O

nearest known ligand 0.73

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.73
CLEC4M Q9H2X3 1/20 0.60
MAPT P10636 1/20 0.58
CYP1A2 P05177 1/20 0.53
CYP3A4 P08684 1/20 0.53
CYP2C19 P33261 1/20 0.53
MEN1 O00255 2/20 0.52
KMT2A Q03164 2/20 0.52
GABRA1 P14867 3/20 0.49
GABRB2 P47870 3/20 0.49
GABRB1 P18505 2/20 0.48
GABRA3 P34903 2/20 0.48
ALDH1A1 P00352 1/20 0.42
TP53 P04637 1/20 0.42
HPGD P15428 1/20 0.42
HSD17B10 Q99714 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7225478 0.85 CLEC4M (0.66) KDM4ECLEC4MMAPTCYP1A2CYP3A4
SCHEMBL4742144 0.84 KDM4E (1.00) KDM4ECLEC4MMAPTCYP1A2CYP3A4
SCHEMBL2660023 0.81 CYP1A2 (0.57) KDM4EMAPTCYP1A2MEN1KMT2A
SCHEMBL9635290 0.79 CYP1A2 (0.66) KDM4ECLEC4MMAPTCYP1A2CYP3A4
SCHEMBL29376920 0.79 CYP1A2 (0.66) KDM4ECLEC4MMAPTCYP1A2CYP3A4
SCHEMBL25208357 0.78 CLEC4M (0.63) KDM4ECLEC4MMAPTCYP1A2CYP3A4
SCHEMBL1353417 0.78 KDM4E (0.61) KDM4ECLEC4MMAPTCYP1A2CYP3A4
SCHEMBL1126279 0.78 CLEC4M (0.78) KDM4ECLEC4MMAPTCYP1A2CYP3A4
SCHEMBL4743455 0.77 MEN1 (0.67) KDM4ECLEC4MMAPTCYP1A2CYP3A4
SCHEMBL29145962 0.77 CLEC4M (0.62) KDM4ECLEC4MMAPTCYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004043930-A1 QUINOLINE DERIVATIVES WHICH ENHANCE COGNITION VIA THE GABA-A RECEPTOR MERCK SHARP & DOHME LIMITED (GB) 2004-05-27 WO disclosed