SCHEMBL2661995

SCHEMBL2661995

Cc1ccc(NC(=O)Nc2ncc(CC(=O)O)s2)c(OCC(C)C)c1.Cc1ccc(NC(=O)Nc2ncc(CC(N)=O)s2)c(OCC(C)C)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 1/20 0.39
ITGA4 P13612 1/20 0.39
ALDH1A1 P00352 1/20 0.37
TSHR P16473 1/20 0.37
LPAR1 Q92633 2/20 0.37
EP300 Q09472 2/20 0.36
MYC P01106 2/20 0.36
MAX P61244 2/20 0.36
OGA O60502 1/20 0.35
CPT1A P50416 1/20 0.35
CPT1B Q92523 1/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
LMNA P02545 1/20 0.35
MAPT P10636 1/20 0.35
MAPK1 P28482 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
MAPK14 Q16539 2/20 0.35
MAPK13 O15264 1/20 0.35
CCNE1 P24864 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1343187 0.96 LPAR1 (0.39) ALDH1A1TSHRLPAR1EP300MYC
SCHEMBL1342497 0.95 ITGB1 (0.42) ITGB1ITGA4ALDH1A1TSHRLPAR1
SCHEMBL1343247 0.86 ITGB1 (0.37) ITGB1ITGA4ALDH1A1TSHRLPAR1
SCHEMBL1342668 0.86 LPAR1 (0.39) ALDH1A1TSHRLPAR1MYCMAX
SCHEMBL1343714 0.85 LPAR1 (0.38) LPAR1EP300MYCMAXMEN1
SCHEMBL1342817 0.85 ADRB2 (0.40) ITGB1ITGA4LPAR1MYCMAX
SCHEMBL1340678 0.84 ITGB1 (0.41) ITGB1ITGA4ALDH1A1LPAR1MYC
SCHEMBL6695295 0.84 AURKA (0.40) LPAR1MAPK14MAPK13CDK2
SCHEMBL1343242 0.84 LPAR1 (0.37) LPAR1EP300MYCMAXMEN1
SCHEMBL1342849 0.83 LPAR1 (0.39) ALDH1A1LPAR1MYCMAXMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1531815-A1 GLUCOKINASE ACTIVATORS NOVO NORDISK A/S (DK) 2005-05-25 EP disclosed
WO-2004002481-A1 ARYL CARBONYL DERIVATIVES AS THERAPEUTIC AGENTS NOVO NORDISK A/S (DK) 2004-01-08 WO disclosed