SCHEMBL2662277

SCHEMBL2662277

O=S(=O)(Oc1cc(O)c2ccccc2c1)C(F)(F)F.Oc1cc(-c2ccc(OC(F)(F)F)cc2)cc2ccccc12

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 1/20 0.48
TPX2 Q9ULW0 1/20 0.48
AKR1C2 P52895 1/20 0.40
AKR1C1 Q04828 1/20 0.40
MMP3 P08254 1/20 0.40
ACP1 P24666 1/20 0.38
CYP11B1 P15538 1/20 0.38
CYP11B2 P19099 1/20 0.38
HSD17B1 P14061 3/20 0.38
HSD17B2 P37059 3/20 0.38
ESR1 P03372 1/20 0.38
ESR2 Q92731 1/20 0.38
PTPN1 P18031 2/20 0.38
PTPRC P08575 1/20 0.38
PTPN2 P17706 1/20 0.38
PTPN6 P29350 1/20 0.38
PTPN9 P43378 1/20 0.38
DUSP3 P51452 1/20 0.38
PTPN11 Q06124 1/20 0.38
PTPN22 Q9Y2R2 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2656803 0.87 AURKA (0.50) AURKATPX2AKR1C2AKR1C1MMP3
SCHEMBL2654823 0.85 NQO2 (0.49) HSD17B1HSD17B2ESR1ESR2PTPN1
SCHEMBL14506126 0.72 CA2 (0.54) HSD17B1HSD17B2ESR1ESR2
SCHEMBL10041706 0.72 CA2 (0.54) HSD17B1HSD17B2ESR1ESR2
SCHEMBL14506139 0.72 CA2 (0.47) CYP11B1CYP11B2ESR1ESR2PTPN1
SCHEMBL25040047 0.72 CA2 (0.47) CYP11B1CYP11B2ESR1ESR2PTPN1
SCHEMBL31538684 0.72 CA2 (0.47) CYP11B1CYP11B2ESR1ESR2PTPN1
SCHEMBL12107241 0.71 CA1 (0.47) AKR1C2PTPN1
SCHEMBL15998741 0.71 HTT (0.39) PTPN1PTGER4
SCHEMBL7154183 0.70 CISD1 (0.51) PTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1863755-A1 SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES Merck & Co., Inc. (US) 2007-12-12 EP disclosed
WO-2006102067-A1 SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES MERCK & CO., INC. (US) 2006-09-28 WO disclosed