SCHEMBL2662867

SCHEMBL2662867

Fc1cc(Br)ccc1-c1cc(-c2ccc(Cl)cc2)[nH]c1-c1ccncc1

nearest known ligand 0.73

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
GCGR P47871 15/20 0.73
MAPK14 Q16539 13/20 0.73
KDM4E B2RXH2 1/20 0.61
ALDH1A1 P00352 1/20 0.61
CYP3A4 P08684 1/20 0.61
MAPT P10636 1/20 0.61
HPGD P15428 1/20 0.61
ALOX15 P16050 1/20 0.61
HSD17B10 Q99714 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2662945 0.84 GCGR (1.00) GCGRMAPK14KDM4EALDH1A1CYP3A4
SCHEMBL2662944 0.81 GCGR (0.60) GCGRMAPK14
SCHEMBL2646773 0.80 GCGR (1.00) GCGRMAPK14
SCHEMBL28643906 0.78 GCGR (0.68) GCGRMAPK14KDM4EALDH1A1CYP3A4
SCHEMBL29691553 0.76 GCGR (1.00) GCGRMAPK14KDM4EALDH1A1CYP3A4
SCHEMBL6362882 0.76 GCGR (1.00) GCGRMAPK14KDM4EALDH1A1CYP3A4
SCHEMBL2645507 0.75 GCGR (0.88) GCGRMAPK14
SCHEMBL2662940 0.74 GCGR (0.97) GCGRMAPK14
SCHEMBL8857820 0.72 ALOX5AP (0.46) GCGRMAPK14ALDH1A1MAPTHPGD
SCHEMBL2658421 0.72 IMPDH2 (0.49) GCGRMAPK14CYP3A4MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997016442-A1 SUBSTITUTED PYRIDYL PYRROLES, COMPOSITIONS CONTAINING SUCH COMPOUNDS AND METHODS OF USE MERCK & CO., INC. (US) 1997-05-09 WO disclosed