SCHEMBL266376

SCHEMBL266376

CN(CCN1CCC(OC(=O)Nc2ccccc2-c2ccccc2)CC1)C(=O)c1ccc(C(=O)NCCN)o1

nearest known ligand 0.64

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 1/20 0.64
CHRM3 P20309 19/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL266143 0.88 CHRM2 (0.71) CHRM2CHRM3
SCHEMBL268975 0.87 CHRM2 (0.66) CHRM2CHRM3
SCHEMBL265206 0.86 CHRM2 (0.64) CHRM2CHRM3
SCHEMBL266133 0.86 CHRM3 (0.62) CHRM2CHRM3
SCHEMBL264846 0.86 CHRM3 (0.61) CHRM2CHRM3
SCHEMBL266375 0.85 CHRM3 (0.64) CHRM3
SCHEMBL265792 0.84 CHRM2 (0.61) CHRM2CHRM3
SCHEMBL274909 0.84 CHRM3 (0.68) CHRM2CHRM3
SCHEMBL265589 0.84 CHRM2 (0.65) CHRM2CHRM3
SCHEMBL644529 0.84 CHRM2 (0.64) CHRM2CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 22 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20060205778-A1 Biphenyl compounds useful as muscarinic receptor antagonists THERAVANCE, INC. 2006-09-14 US claimed
CN-104642793-A Reserve cow feed with low-phosphorous emission UNIV ZHEJIANG 2015-05-27 CN disclosed
US-20130274288-A1 BIPHENYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS THERAVANCE, INC. (US) 2013-10-17 US disclosed
US-8487107-B2 Biphenyl compounds useful as muscarinic receptor antagonists THERAVANCE, INC. (US) 2013-07-16 US disclosed
US-8377966-B2 Biphenyl compounds useful as muscarinic receptor antagonists THERAVANCE, INC. (US) 2013-02-19 US disclosed
US-20120122926-A1 BIPHENYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS THERAVANCE, INC. (US) 2012-05-17 US disclosed
US-8133905-B2 Biphenyl compounds useful as muscarinic receptor antagonists THERAVANCE, INC. (US) 2012-03-13 US disclosed
US-8124627-B2 Biphenyl compounds useful as muscarinic receptor antagonists THERAVANCE, INC. (US) 2012-02-28 US disclosed
US-7790923-B2 Process for the production of phosphorous compounds BASF Nederland B.V. and University of Amsterdam (US) 2010-09-07 US disclosed
US-20100125079-A1 BIPHENYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS THERAVANCE, INC. (US) 2010-05-20 US disclosed
US-20100056541-A1 BIPHENYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS THERAVANCE, INC. (US) 2010-03-04 US disclosed
US-7659403-B2 Bronchodilators; treating chronic obstructive pulmonary disease or asthma; long duration of action; reduced side effects, such as dry-mouth and constipation; e.g. biphenyl-2-ylcarbamic acid 1-(2-[methyl(3-(2-[(thiophen-2-ylmethyl)amino]ethylcarbamoyl)benzoyl)amino]ethyl)piperidin-4-yl ester THERAVANCE, INC. (US) 2010-02-09 US disclosed
US-7632847-B2 Bronchodilators; treating chronic obstructive pulmonary disease or asthma; long duration of action; reduced side effects, such as dry-mouth and constipation; e.g. biphenyl-2-ylcarbamic acid 1-(2-(3-[3-(4-hydroxybenzylamino)propionylamino]benzoylamino)ethyl)piperidin-4-yl ester THERAVANCE, INC. (US) 2009-12-15 US disclosed
US-20090082595-A1 Process for the production of phosphorous compounds ENGELHARD DE MEERN B.V. (NL) 2009-03-26 US disclosed
EP-1987045-A1 PROCESS FOR THE PRODUCTION OF PHOSPHOROUS COMPOUNDS Engelhard De Meern B.V. (NL) 2008-11-05 EP disclosed
EP-1816132-A1 Process for the production of phosphorous compounds ENGELHARD CORPORATION (US) 2007-08-08 EP disclosed
WO-2007086745-A1 PROCESS FOR THE PRODUCTION OF PHOSPHOROUS COMPOUNDS ENGELHARD DE MEERN B.V. (NL) 2007-08-02 WO disclosed
US-20060205784-A1 Biphenyl compounds useful as muscarinic receptor antagonists THERAVANCE, INC. 2006-09-14 US disclosed
US-20060205778-A1 Biphenyl compounds useful as muscarinic receptor antagonists THERAVANCE, INC. 2006-09-14 US disclosed
US-20060205777-A1 Biphenyl compounds useful as muscarinic receptor antagonists THERAVANCE, INC. 2006-09-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100056541-A1 BIPHENYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS CHRM2, CHRM1, CHRM3 CHRM2 1/4885CHRM3 3/4885
US-20060205778-A1 Biphenyl compounds useful as muscarinic receptor antagonists CHRM2, CHRM1, CHRM3 CHRM2 1/4885CHRM3 3/4885
US-20060205784-A1 Biphenyl compounds useful as muscarinic receptor antagonists CHRM2, CHRM1, CHRM3 CHRM2 1/4885CHRM3 3/4885
US-20060205777-A1 Biphenyl compounds useful as muscarinic receptor antagonists CHRM2, CHRM1, CHRM3 CHRM2 1/4885CHRM3 3/4885
US-20130274288-A1 BIPHENYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS CHRM2, CHRM1, CHRM3 CHRM2 1/4885CHRM3 3/4885
US-20100125079-A1 BIPHENYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS CHRM2, CHRM1, CHRM3 CHRM2 1/4885CHRM3 3/4885
US-20120122926-A1 BIPHENYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS CHRM2, CHRM1, CHRM3 CHRM2 1/4885CHRM3 3/4885
US-20090082595-A1 Process for the production of phosphorous compounds TPMT, NUDT1, MTAP CHRM2 4594/4885CHRM3 4728/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.