SCHEMBL26645016

SCHEMBL26645016

COc1ccc(-c2nn3c(c2-c2ccncc2)CN(C(=O)OC(C)(C)C)CC3)cc1F

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CSNK1E P49674 9/20 0.42
CFTR P13569 1/20 0.42
CSNK1D P48730 6/20 0.41
GALR2 O43603 1/20 0.39
GALR1 P47211 1/20 0.39
KDM1A O60341 1/20 0.39
SMPD3 Q9NY59 2/20 0.38
GPR119 Q8TDV5 2/20 0.38
ABHD6 Q9BV23 1/20 0.38
PDE4A P27815 2/20 0.37
PDE4B Q07343 2/20 0.37
PDE4C Q08493 1/20 0.37
PDE4D Q08499 1/20 0.37
CYP17A1 P05093 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30622850 1.00 CSNK1E (0.42) CSNK1ECFTRCSNK1DGALR2GALR1
SCHEMBL26645587 0.90 CFTR (0.42) CSNK1ECFTRCSNK1DSMPD3GPR119
SCHEMBL30622740 0.90 CFTR (0.42) CSNK1ECFTRCSNK1DSMPD3GPR119
SCHEMBL26645275 0.89 CSNK1E (0.43) CSNK1ECSNK1DGPR119PDE4APDE4B
SCHEMBL30622919 0.88 CSNK1E (0.46) CSNK1ECSNK1DGPR119
SCHEMBL26645204 0.88 CSNK1E (0.46) CSNK1ECSNK1DGPR119
SCHEMBL26645681 0.86 CSNK1E (0.48) CSNK1ECSNK1DGPR119
SCHEMBL30622425 0.86 CSNK1E (0.42) CSNK1ECSNK1DKDM1APDE4APDE4B
SCHEMBL26644880 0.86 CSNK1E (0.42) CSNK1ECSNK1DKDM1APDE4APDE4B
SCHEMBL30623018 0.85 CSNK1E (0.44) CSNK1ECFTRCSNK1DGALR2GALR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023213882-A1 IRREVERSIBLE MUTEGFR INHIBITORS BAYER AKTIENGESELLSCHAFT (DE) 2023-11-09 WO disclosed