SCHEMBL26645587

SCHEMBL26645587

COc1ccc(-c2nn3c(c2-c2ccncc2)CN(C(=O)OC(C)(C)C)CC3)cc1Cl

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CFTR P13569 2/20 0.42
CSNK1E P49674 2/20 0.41
CSNK1D P48730 1/20 0.41
PGK1 P00558 1/20 0.39
PDE4A P27815 1/20 0.39
PDE4B Q07343 1/20 0.39
PDE4C Q08493 1/20 0.39
PDE4D Q08499 1/20 0.39
MAPK14 Q16539 5/20 0.39
SMPD3 Q9NY59 2/20 0.38
SUV39H2 Q9H5I1 4/20 0.38
CACNB4 O00305 2/20 0.38
CACNA1A O00555 2/20 0.38
CACNA1G O43497 2/20 0.38
CACNG3 O60359 2/20 0.38
CACNA1F O60840 2/20 0.38
CACNA1H O95180 2/20 0.38
CACNB3 P54284 2/20 0.38
CACNA2D1 P54289 2/20 0.38
CACNG7 P62955 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30622740 1.00 CFTR (0.42) CFTRCSNK1ECSNK1DPGK1PDE4A
SCHEMBL26645014 0.91 CSNK1E (0.43) CSNK1ECSNK1DGPR119
SCHEMBL30622825 0.91 CSNK1E (0.43) CSNK1ECSNK1DGPR119
SCHEMBL26645016 0.90 CSNK1E (0.42) CFTRCSNK1ECSNK1DPDE4APDE4B
SCHEMBL30622850 0.90 CSNK1E (0.42) CFTRCSNK1ECSNK1DPDE4APDE4B
SCHEMBL26645805 0.88 CSNK1E (0.42) CSNK1ECSNK1DGPR119
SCHEMBL26645275 0.87 CSNK1E (0.43) CSNK1ECSNK1DPDE4APDE4BPDE4C
SCHEMBL30622922 0.86 CSNK1E (0.43) CSNK1ECSNK1DMAPK14
SCHEMBL26645443 0.86 CSNK1E (0.43) CSNK1ECSNK1DMAPK14
SCHEMBL26645019 0.86 CSNK1D (0.47) CSNK1ECSNK1DMAPK14CACNB4CACNA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023213882-A1 IRREVERSIBLE MUTEGFR INHIBITORS BAYER AKTIENGESELLSCHAFT (DE) 2023-11-09 WO disclosed